SCHEMBL22702017

SCHEMBL22702017

CS(=O)(=O)N1CCC(N/C=C\NN)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.41
EPHX2 P34913 3/20 0.38
KDM1A O60341 1/20 0.38
EPHX1 P07099 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
FABP6 P51161 1/20 0.38
LMNA P02545 1/20 0.36
ALDH1A1 P00352 2/20 0.35
SMYD3 Q9H7B4 1/20 0.35
TSHR P16473 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MAPT P10636 1/20 0.34
IDO1 P14902 1/20 0.34
POLB P06746 1/20 0.33
CYP2C19 P33261 1/20 0.33
CCNE2 O96020 1/20 0.33
CDK4 P11802 1/20 0.33
CCND1 P24385 1/20 0.33
CCNE1 P24864 1/20 0.33
CDK2 P24941 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22702143 0.84 TP53 (0.42) TP53EPHX2KDM1AEPHX1NPSR1
SCHEMBL774350 0.78 ADH1B (0.50) TP53EPHX2KDM1AEPHX1NPSR1
SCHEMBL29259766 0.77 TP53 (0.48) TP53EPHX2KDM1AEPHX1NPSR1
SCHEMBL18375610 0.71
SCHEMBL5344959 0.71 TP53 (0.50) TP53EPHX2KDM1AEPHX1NPSR1
SCHEMBL12820051 0.70 TP53 (0.48) TP53EPHX2KDM1AEPHX1NPSR1
SCHEMBL773447 0.68 ADH1B (0.41) TP53EPHX2KDM1AEPHX1NPSR1
SCHEMBL21746087 0.68 TP53 (0.41) TP53EPHX2KDM1AEPHX1NPSR1
SCHEMBL20609817 0.67 TP53 (0.46) TP53EPHX2KDM1AEPHX1NPSR1
SCHEMBL12404039 0.67 TP53 (0.46) TP53EPHX2KDM1AEPHX1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3319955-B1 6-AMINO-QUINOLINE-3-CARBONITRILS AS COT MODULATORS GILEAD SCIENCES INC (US) 2020-11-25 EP disclosed