SCHEMBL22709208

SCHEMBL22709208

CN(C=O)CCN(C)C(=O)C(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 1/20 0.37
USP2 O75604 1/20 0.34
ALOX15 P16050 1/20 0.34
MEN1 O00255 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
KMT2A Q03164 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CTSK P43235 3/20 0.32
BRD4 O60885 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27043895 0.84 RIPK1 (0.44) RIPK1MEN1CYP3A4CYP2C9CYP2C19
SCHEMBL8137111 0.78 RIPK1 (0.41) RIPK1MEN1CYP3A4CYP2C9CYP2C19
SCHEMBL24476085 0.76 RIPK1 (0.40) RIPK1MEN1CYP3A4CYP2C9CYP2C19
SCHEMBL15434422 0.76 USP2 (0.38) USP2ALOX15
SCHEMBL12392730 0.74 KDM4E (0.46) RIPK1MEN1CYP3A4CYP2C9CYP2C19
SCHEMBL9814035 0.74 TSHR (0.47) USP2ALOX15
SCHEMBL28551868 0.73 BRD4 (0.37) RIPK1MEN1CYP3A4CYP2C9CYP2C19
SCHEMBL9010937 0.73 RIPK1 (0.37) RIPK1MEN1CYP3A4CYP2C9CYP2C19
SCHEMBL1712608 0.73 MAPT (0.46) RIPK1ALOX15MEN1CYP3A4CYP2C9
SCHEMBL1712606 0.73 RIPK1 (0.37) RIPK1MEN1CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020236825-A2 MCL-1 INHIBITOR ANTIBODY-DRUG CONJUGATES AND METHODS OF USE NOVARTIS AG (CH) 2020-11-26 WO disclosed