SCHEMBL22720104

SCHEMBL22720104

Nc1cc(F)ccc1C(=O)NC1CCCC1

nearest known ligand 0.60

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.60
NPC1 O15118 11/20 0.56
RAB9A P51151 10/20 0.56
ALDH1A1 P00352 4/20 0.54
KMT2A Q03164 1/20 0.54
ATM Q13315 1/20 0.53
MLLT1 Q03111 1/20 0.52
SMN1; SMN2 Q16637 2/20 0.51
KDM1A O60341 1/20 0.51
MAOA P21397 1/20 0.51
POLB P06746 1/20 0.49
CNR1 P21554 2/20 0.48
CNR2 P34972 2/20 0.48
TDP1 Q9NUW8 1/20 0.48
HTR2B P41595 1/20 0.48
KDM4E B2RXH2 1/20 0.48
LMNA P02545 1/20 0.48
HTT P42858 1/20 0.48
MAPT P10636 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22720134 0.98 NPC1 (0.59) HPGDNPC1RAB9AALDH1A1KMT2A
SCHEMBL13161899 0.87 HPGD (0.56) HPGDNPC1RAB9AALDH1A1KMT2A
SCHEMBL22720149 0.87 NPC1 (0.59) HPGDNPC1RAB9AALDH1A1KMT2A
SCHEMBL22720107 0.82 RAB9A (0.68) HPGDNPC1RAB9AALDH1A1KMT2A
SCHEMBL6367825 0.81 HPGD (0.63) HPGDNPC1RAB9AALDH1A1KMT2A
SCHEMBL7985363 0.81 HPGD (0.63) HPGDNPC1RAB9AALDH1A1KMT2A
SCHEMBL26170042 0.81 NPC1 (0.56) HPGDNPC1RAB9AALDH1A1KMT2A
SCHEMBL22720141 0.81 NPC1 (0.70) HPGDNPC1RAB9AALDH1A1KMT2A
SCHEMBL22720169 0.79 RAB9A (0.63) HPGDNPC1RAB9AALDH1A1KMT2A
SCHEMBL13498283 0.79 CRBN (0.57) HPGDNPC1RAB9AALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020239050-A1 2-(2-CHLORO-4-METHYLPHENYL)QUINAZOLINE-4(3H)-KETONE COMPOUND AND MEDICAL USE THEREOF 中国人民解放军军事科学院军事医学研究院 2020-12-03 WO disclosed
CN-110041272-B 2- (2-chlorphenyl) quinazoline-4 (3H) -ketone derivative and preparation method and application thereof 中国人民解放军军事科学院军事医学研究院 2020-10-30 CN disclosed
CN-110041273-B 2- (2-chloro-4-methylphenyl) quinazoline-4 (3H) -ketone compound and medical application thereof 中国人民解放军军事科学院军事医学研究院 2020-10-20 CN disclosed
CN-110041273-A 2- (the chloro- 4- aminomethyl phenyl of 2-) quinazoline -4 (3H) -one class compound and its medical usage 中国人民解放军军事科学院军事医学研究院 2019-07-23 CN disclosed
CN-110041272-A 2- (2- chlorphenyl) quinazoline -4 (3H) -one analog derivative and its preparation method and application 中国人民解放军军事科学院军事医学研究院 2019-07-23 CN disclosed