SCHEMBL22720133

SCHEMBL22720133

COc1ccc2c(=O)n(C3CCCC3)c(-c3ccc(C)cc3Cl)nc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 5/20 0.46
KCNH2 Q12809 4/20 0.46
CRHR1 P34998 1/20 0.45
TSHR P16473 2/20 0.43
PLA2G1B P04054 1/20 0.43
HSD17B10 Q99714 1/20 0.43
ATG4B Q9Y4P1 1/20 0.43
PIK3CA P42336 5/20 0.43
MPI P34949 1/20 0.42
ALOX15 P16050 2/20 0.41
GAA P10253 1/20 0.41
PRKACA P17612 1/20 0.40
RPS6KB1 P23443 1/20 0.40
GSK3B P49841 1/20 0.40
ROCK1 Q13464 1/20 0.40
CYP1A1 P04798 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP1B1 Q16678 1/20 0.39
PRKDC P78527 1/20 0.39
MTOR P42345 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22720176 0.90 ALOX15 (0.46) TSHRPLA2G1BHSD17B10ATG4BPIK3CA
SCHEMBL22736786 0.89 ALOX15 (0.48) TSHRPLA2G1BHSD17B10ATG4BPIK3CA
SCHEMBL22720084 0.88 GAA (0.43) HRH3KCNH2TSHRPLA2G1BHSD17B10
SCHEMBL22720110 0.86 TSHR (0.40) CRHR1TSHRPLA2G1BHSD17B10ATG4B
SCHEMBL22720123 0.85 GAA (0.42) HRH3KCNH2TSHRPLA2G1BHSD17B10
SCHEMBL22720130 0.84 ALOX15 (0.44) HRH3KCNH2TSHRPLA2G1BHSD17B10
SCHEMBL22720124 0.84 GAA (0.59) TSHRALOX15GAAALDH1A1KDM4E
SCHEMBL22720187 0.84 GAA (0.46) TSHRHSD17B10PIK3CAALOX15GAA
SCHEMBL22720121 0.83 GAA (0.61) TSHRALOX15GAAALDH1A1KDM4E
SCHEMBL22720182 0.83 GAA (0.61) TSHRALOX15GAAALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020239050-A1 2-(2-CHLORO-4-METHYLPHENYL)QUINAZOLINE-4(3H)-KETONE COMPOUND AND MEDICAL USE THEREOF 中国人民解放军军事科学院军事医学研究院 2020-12-03 WO disclosed
WO-2020239050-A1 2-(2-CHLORO-4-METHYLPHENYL)QUINAZOLINE-4(3H)-KETONE COMPOUND AND MEDICAL USE THEREOF 中国人民解放军军事科学院军事医学研究院 2020-12-03 WO disclosed