SCHEMBL22720172

SCHEMBL22720172

Nc1c(C(=O)Nc2ccccc2)cccc1C(F)(F)F

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 3/20 0.66
KCNK3 O14649 3/20 0.62
KCNK9 Q9NPC2 3/20 0.62
RXFP1 Q9HBX9 2/20 0.53
F2R P25116 1/20 0.52
ATR Q13535 1/20 0.52
ALDH1A1 P00352 2/20 0.51
LMNA P02545 4/20 0.50
P2RX1 P51575 2/20 0.50
MEN1 O00255 2/20 0.50
HPGD P15428 2/20 0.50
KMT2A Q03164 2/20 0.50
KDM4E B2RXH2 1/20 0.50
TP53 P04637 1/20 0.50
HTT P42858 1/20 0.50
HSD17B10 Q99714 1/20 0.50
PRKCI P41743 1/20 0.50
GAA P10253 2/20 0.49
POLB P06746 1/20 0.49
TDP1 Q9NUW8 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27463747 0.88 PTGS1 (0.55) PTGS1KCNK3KCNK9ATRALDH1A1
SCHEMBL5332281 0.85 KCNK3 (0.75) PTGS1KCNK3KCNK9RXFP1F2R
SCHEMBL7213018 0.83 KCNK3 (0.63) PTGS1KCNK3KCNK9RXFP1F2R
SCHEMBL734924 0.80 CYP1A2 (0.59) PTGS1RXFP1ALDH1A1HPGDKDM4E
SCHEMBL678924 0.80 PTGS1 (0.72) PTGS1KCNK3KCNK9RXFP1F2R
SCHEMBL2061662 0.80 GAA (0.49) PTGS1KCNK3KCNK9LMNAGAA
SCHEMBL392794 0.79 ALDH1A1 (0.59) PTGS1ALDH1A1LMNAMEN1HPGD
SCHEMBL357846 0.79 PTGS1 (0.55) PTGS1KCNK3KCNK9ATRALDH1A1
SCHEMBL11583305 0.79 KCNK3 (0.58) PTGS1KCNK3KCNK9RXFP1F2R
SCHEMBL28799328 0.79 PTGS1 (0.62) PTGS1KCNK3KCNK9RXFP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020239050-A1 2-(2-CHLORO-4-METHYLPHENYL)QUINAZOLINE-4(3H)-KETONE COMPOUND AND MEDICAL USE THEREOF 中国人民解放军军事科学院军事医学研究院 2020-12-03 WO disclosed
CN-110041273-B 2- (2-chloro-4-methylphenyl) quinazoline-4 (3H) -ketone compound and medical application thereof 中国人民解放军军事科学院军事医学研究院 2020-10-20 CN disclosed
CN-110041273-A 2- (the chloro- 4- aminomethyl phenyl of 2-) quinazoline -4 (3H) -one class compound and its medical usage 中国人民解放军军事科学院军事医学研究院 2019-07-23 CN disclosed