SCHEMBL22720307

SCHEMBL22720307

Cc1c(Br)nc(OCC2CCCN2C)nc1N1CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KRAS P01116 12/20 0.42
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
MEN1 O00255 1/20 0.36
MAPT P10636 1/20 0.36
TSHR P16473 1/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
GPR119 Q8TDV5 1/20 0.36
CHRNB2 P17787 1/20 0.36
CHRNA4 P43681 1/20 0.36
OPRM1 P35372 1/20 0.36
OPRD1 P41143 1/20 0.36
OGFRL1 Q5TC84 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22724618 1.00 KRAS (0.42) KRASCHRNB4CHRNA3MEN1MAPT
SCHEMBL30957839 1.00 KRAS (0.42) KRASCHRNB4CHRNA3MEN1MAPT
SCHEMBL22720285 0.89 KRAS (0.42) KRASCHRNB4CHRNA3GPR119CHRNB2
SCHEMBL22720353 0.88 KRAS (0.44) KRASCHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL22720351 0.88 KRAS (0.44) KRASCHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL22720294 0.85 KRAS (0.56) KRAS
SCHEMBL22720296 0.85 KRAS (0.56) KRAS
SCHEMBL22720271 0.84 KRAS (0.46) KRASCHRNB4CHRNA3GPR119CHRNB2
SCHEMBL22720227 0.84 KRAS (0.46) KRASCHRNB4CHRNA3GPR119CHRNB2
SCHEMBL30957849 0.84 KRAS (0.46) KRASCHRNB4CHRNA3GPR119CHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113396147-B Aromatic heterocyclic derivative regulator, preparation method and application thereof 上海翰森生物医药科技有限公司 2024-06-18 CN disclosed
WO-2020239123-A1 AROMATIC HETEROCYCLIC DERIVATIVE MODULATOR AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海翰森生物医药科技有限公司 2020-12-03 WO disclosed