SCHEMBL22720285

SCHEMBL22720285

Cc1nc(OC[C@@H]2CCCN2C)nc(N2CCN(C(=O)OC(C)(C)C)CC2)c1Br

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KRAS P01116 13/20 0.42
CHRNB4 P30926 2/20 0.38
CHRNA3 P32297 2/20 0.38
KCNH2 Q12809 1/20 0.37
GPR119 Q8TDV5 1/20 0.36
CHRNB2 P17787 2/20 0.36
CHRNA4 P43681 2/20 0.36
CHRNB1 P11230 1/20 0.36
CHRNB3 Q05901 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30957839 0.89 KRAS (0.42) KRASCHRNB4CHRNA3GPR119CHRNB2
SCHEMBL22724618 0.89 KRAS (0.42) KRASCHRNB4CHRNA3GPR119CHRNB2
SCHEMBL22720307 0.89 KRAS (0.42) KRASCHRNB4CHRNA3GPR119CHRNB2
SCHEMBL28538875 0.88 KRAS (0.44) KRASCHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL28538876 0.88 KRAS (0.44) KRASCHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL22720272 0.87 KRAS (0.43) KRASCHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL22720271 0.84 KRAS (0.46) KRASCHRNB4CHRNA3GPR119CHRNB2
SCHEMBL30957849 0.84 KRAS (0.46) KRASCHRNB4CHRNA3GPR119CHRNB2
SCHEMBL22720227 0.84 KRAS (0.46) KRASCHRNB4CHRNA3GPR119CHRNB2
SCHEMBL22720268 0.84 KRAS (0.39) KRASGPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020239123-A1 AROMATIC HETEROCYCLIC DERIVATIVE MODULATOR AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海翰森生物医药科技有限公司 2020-12-03 WO disclosed