SCHEMBL22720571

SCHEMBL22720571

c1ccc(CN2CCc3c(nc(-c4ccccc4)nc3-c3ccccc3)C2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.48
MEN1 O00255 2/20 0.48
PARP1 P09874 1/20 0.47
TNKS2 Q9H2K2 1/20 0.47
PARP2 Q9UGN5 1/20 0.47
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
GLA P06280 1/20 0.46
GAA P10253 1/20 0.46
MAPT P10636 1/20 0.46
HPGD P15428 1/20 0.46
CFTR P13569 6/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
C5AR1 P21730 1/20 0.45
LMNA P02545 1/20 0.45
ACHE P22303 1/20 0.45
CYP2D6 P10635 1/20 0.45
KCNH2 Q12809 1/20 0.45
SLC6A5 Q9Y345 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5999914 0.88 KMT2A (0.54) KMT2AMEN1PARP1TNKS2PARP2
SCHEMBL4147065 0.86 C5AR1 (0.57) KMT2AMEN1PARP1TNKS2PARP2
SCHEMBL183618 0.85 P2RX7 (0.53) KMT2AMEN1PARP1TNKS2PARP2
SCHEMBL16034465 0.85 KMT2A (0.53) KMT2AMEN1PARP1TNKS2PARP2
SCHEMBL183455 0.84 HTR2A (0.51) KMT2AMEN1PARP1TNKS2PARP2
Hydrochloric Acid SCHEMBL6298078 0.84 P2RX7 (0.52) KMT2AMEN1PARP1TNKS2PARP2
SCHEMBL183374 0.82 PARP1 (0.46) KMT2AMEN1PARP1TNKS2PARP2
SCHEMBL12386805 0.81 P2RX7 (0.50) KMT2AMEN1PARP1TNKS2PARP2
SCHEMBL22720440 0.80 KMT2A (0.49) KMT2AMEN1PARP1TNKS2PARP2
SCHEMBL183675 0.77 HTR2A (0.64) KMT2AMEN1PARP1TNKS2PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020239077-A1 NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVE REGULATOR, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 上海翰森生物医药科技有限公司 2020-12-03 WO disclosed