SCHEMBL22729474

SCHEMBL22729474

Cc1cn(C)c(=O)c2c(C(=O)NC3CCCCC3NC(=O)OC(C)(C)C)cn(C)c12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
ALDH1A1 P00352 3/20 0.39
USP2 O75604 2/20 0.36
NPSR1 Q6W5P4 2/20 0.36
MEN1 O00255 1/20 0.36
GAA P10253 1/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
TAS1R3 Q7RTX0 4/20 0.36
TAS1R1 Q7RTX1 4/20 0.36
TAS1R2 Q8TE23 4/20 0.36
POLB P06746 1/20 0.35
SYK P43405 1/20 0.34
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
LMNA P02545 1/20 0.34
TSHR P16473 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23139760 1.00 HDAC4 (0.39) HDAC4HDAC6ALDH1A1USP2NPSR1
SCHEMBL23139207 1.00 HDAC4 (0.39) HDAC4HDAC6ALDH1A1USP2NPSR1
SCHEMBL23139740 1.00 HDAC4 (0.39) HDAC4HDAC6ALDH1A1USP2NPSR1
SCHEMBL23139724 1.00 HDAC4 (0.39) HDAC4HDAC6ALDH1A1USP2NPSR1
SCHEMBL22729446 0.87 ALDH1A1 (0.40) ALDH1A1USP2NPSR1MEN1GAA
SCHEMBL22729612 0.87 ALDH1A1 (0.40) ALDH1A1USP2NPSR1MEN1GAA
SCHEMBL22729728 0.87 ALDH1A1 (0.40) ALDH1A1USP2NPSR1MEN1GAA
SCHEMBL23116405 0.87 ALDH1A1 (0.40) ALDH1A1USP2NPSR1MEN1GAA
SCHEMBL23116406 0.87 ALDH1A1 (0.40) ALDH1A1USP2NPSR1MEN1GAA
SCHEMBL22729602 0.83 ALDH1A1 (0.42) ALDH1A1USP2NPSR1MEN1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3747885-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2020-12-09 EP disclosed