SCHEMBL2273252

SCHEMBL2273252

COC(=O)c1ccc2c(C3CCCCC3)c3n(c2c1)C[C@@H](CCCO)COc1ccccc1-3

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCA P17252 1/20 0.57
MMP12 P39900 1/20 0.57
NR1I2 O75469 5/20 0.37
KCNH2 Q12809 6/20 0.35
SCN9A Q15858 3/20 0.35
CYP3A4 P08684 4/20 0.34
CYP2C9 P11712 2/20 0.34
CYP2C19 P33261 2/20 0.34
ALDH1A1 P00352 2/20 0.33
NPSR1 Q6W5P4 2/20 0.33
SCN5A Q14524 2/20 0.33
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33
KDM4E B2RXH2 1/20 0.33
LMNA P02545 1/20 0.33
HPGD P15428 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL393359 0.92 PRKCA (0.60) PRKCAMMP12NR1I2KCNH2SCN9A
SCHEMBL393360 0.92 PRKCA (0.60) PRKCAMMP12NR1I2KCNH2SCN9A
SCHEMBL394862 0.91 PRKCA (0.58) PRKCAMMP12NR1I2KCNH2SCN9A
SCHEMBL394863 0.91 PRKCA (0.58) PRKCAMMP12NR1I2KCNH2SCN9A
SCHEMBL14110621 0.91 PRKCA (0.57) PRKCAMMP12NR1I2KCNH2SCN9A
SCHEMBL2279970 0.91 PRKCA (0.59) PRKCAMMP12NR1I2KCNH2SCN9A
SCHEMBL4217906 0.90 PRKCA (0.67) PRKCAMMP12NR1I2SCN9ACYP3A4
SCHEMBL2275845 0.88 PRKCA (0.52) PRKCAMMP12NR1I2KCNH2SCN9A
SCHEMBL2275096 0.88 PRKCA (0.57) PRKCAMMP12NR1I2KCNH2SCN9A
SCHEMBL2275820 0.88 PRKCA (0.57) PRKCAMMP12NR1I2KCNH2SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7989438-B2 Therapeutic compounds ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2011-08-02 US disclosed