SCHEMBL22757148

SCHEMBL22757148

COc1ccc(-c2nc(-c3ccc(Nc4ccccc4)cc3)no2)cc1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 3/20 0.78
S1PR1 P21453 1/20 0.78
NPC1 O15118 11/20 0.65
RAB9A P51151 11/20 0.65
MAPT P10636 7/20 0.65
SMN1; SMN2 Q16637 5/20 0.65
NPSR1 Q6W5P4 1/20 0.65
LMNA P02545 1/20 0.63
MEN1 O00255 1/20 0.59
KMT2A Q03164 1/20 0.59
NFKB1 P19838 3/20 0.58
NFKB2 Q00653 3/20 0.58
RELA Q04206 3/20 0.58
TP53 P04637 2/20 0.58
TDP1 Q9NUW8 1/20 0.58
PKM P14618 2/20 0.58
HSP90AA1 P07900 1/20 0.58
L3MBTL1 Q9Y468 1/20 0.58
HAVCR2 Q8TDQ0 1/20 0.55
KDM4E B2RXH2 2/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16592723 0.97 NR1H4 (0.83) NR1H4S1PR1NPC1RAB9AMAPT
SCHEMBL16592612 0.94 RAB9A (0.72) NR1H4S1PR1NPC1RAB9AMAPT
SCHEMBL16592771 0.90 NR1H4 (0.63) NR1H4S1PR1NPC1RAB9AMAPT
SCHEMBL16602947 0.89 NPC1 (0.83) NR1H4S1PR1NPC1RAB9AMAPT
SCHEMBL6697420 0.88 NR1H4 (1.00) NR1H4S1PR1NPC1RAB9AMAPT
SCHEMBL7291752 0.88 NR1H4 (1.00) NR1H4S1PR1NPC1RAB9AMAPT
SCHEMBL16592626 0.86 NPC1 (0.64) NR1H4S1PR1NPC1RAB9AMAPT
SCHEMBL16592746 0.84 NR1H4 (0.65) NR1H4S1PR1NPC1RAB9AMAPT
SCHEMBL1608386 0.84 RAB9A (0.70) NR1H4S1PR1NPC1RAB9AMAPT
SCHEMBL16592774 0.81 S1PR1 (0.70) NR1H4S1PR1NPC1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2853532-B1 1,2,4-oxadiazole derivatives as allosteric modulators of metabotropic glutamate receptors belonging to group III INST FARMAKOLOGII POLSKIEJ AKADEMII NAUK (PL) 2020-12-09 EP disclosed