SCHEMBL22760128

SCHEMBL22760128

CCOC(=O)c1cc2c(Cl)c(F)ccc2n1-c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.51
KMT2A Q03164 3/20 0.51
MAPT P10636 4/20 0.51
TP53 P04637 3/20 0.51
THRB P10828 2/20 0.51
KDM4E B2RXH2 1/20 0.48
ALDH1A1 P00352 2/20 0.47
GAA P10253 1/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
RECQL P46063 1/20 0.46
PTGES O14684 1/20 0.43
MAT2A P31153 1/20 0.43
NPSR1 Q6W5P4 2/20 0.42
SIRT2 Q8IXJ6 1/20 0.42
SIRT1 Q96EB6 1/20 0.42
MAPK1 P28482 1/20 0.42
TSHR P16473 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22760161 0.88 MEN1 (0.53) MEN1KMT2AMAPTTP53THRB
SCHEMBL22760544 0.88 MEN1 (0.53) MEN1KMT2AMAPTTP53THRB
SCHEMBL22760404 0.83 MAPT (0.57) MAPTKDM4EALDH1A1GAASMN1; SMN2
SCHEMBL19332145 0.82 ALDH1A1 (0.44) MAPTKDM4EALDH1A1GAASMN1; SMN2
SCHEMBL22760420 0.79 MAPT (0.47) MEN1KMT2AMAPTTP53THRB
SCHEMBL22760557 0.76 MAPT (0.51) MEN1KMT2AMAPTTP53KDM4E
SCHEMBL22760094 0.75 ALDH1A1 (0.51) MEN1KMT2AMAPTTP53THRB
SCHEMBL8296756 0.75 ALDH1A1 (0.63) MEN1KMT2AMAPTKDM4EALDH1A1
SCHEMBL4699355 0.74 RECQL (0.63) MEN1KMT2AMAPTTP53THRB
SCHEMBL22760095 0.73 MAPT (0.48) MEN1KMT2AMAPTTP53THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020244462-A1 INDOLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF 中国药科大学 2020-12-10 WO disclosed