SCHEMBL22761663

SCHEMBL22761663

O=C(O)c1c(-c2ccccc2F)nc2sccn12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.44
NTRK1 P04629 2/20 0.43
IDO1 P14902 2/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
PTGS2 P35354 5/20 0.40
PTGS1 P23219 2/20 0.39
NLRP3 Q96P20 1/20 0.38
PRKD3 O94806 1/20 0.38
MAP4K4 O95819 1/20 0.38
FGFR1 P11362 1/20 0.38
FRK P42685 1/20 0.38
MAPK8 P45983 1/20 0.38
MAPK9 P45984 1/20 0.38
CSNK1A1 P48729 1/20 0.38
CSNK1D P48730 1/20 0.38
GSK3B P49841 1/20 0.38
CSNK1G2 P78368 1/20 0.38
PRKCD Q05655 1/20 0.38
ERBB4 Q15303 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22761661 0.81 HSD17B10 (0.59) HSD17B10NTRK1IDO1GAAMAPT
SCHEMBL6940612 0.79 MPL (0.43) HSD17B10NTRK1IDO1GAAMAPT
SCHEMBL4716917 0.73 IDO1 (0.69) HSD17B10NTRK1IDO1GAAMAPT
SCHEMBL31468428 0.72 TNK2 (0.41) HSD17B10MAPT
SCHEMBL22761829 0.70 HSD17B10 (0.56) HSD17B10NTRK1IDO1GAAMAPT
SCHEMBL31468331 0.69 MAOA (0.49) HSD17B10LDHA
SCHEMBL27490015 0.69 GAA (0.45) HSD17B10NTRK1IDO1GAAMAPT
SCHEMBL1339567 0.68 DYRK1A (0.56) HSD17B10MAPT
SCHEMBL1340720 0.68 MAPK1 (0.42) HSD17B10
SCHEMBL14953477 0.68 KDM5B (0.39) MAPTPRKD3PRKD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020247445-A1 IMIDAZOLO DERIVATIVES, COMPOSITIONS AND METHODS AS OREXIN ANTAGONISTS HAGER BIOSCIENCES, LLC (US) 2020-12-10 WO disclosed