SCHEMBL22761841

SCHEMBL22761841

FC(F)(F)c1ccc(NC[C@@H]2CCCN2)nc1

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
IL1B P01584 3/20 0.53
IDO1 P14902 3/20 0.52
TDO2 P48775 3/20 0.52
SCN9A Q15858 3/20 0.46
LTA4H P09960 1/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
IRAK4 Q9NWZ3 1/20 0.43
DPP4 P27487 1/20 0.43
CCNT1 O60563 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15173475 0.83 HCRTR1 (0.46)
SCHEMBL296168 0.83 IL1B (0.41) IL1BNPC1RAB9A
SCHEMBL18734317 0.83 HCRTR1 (0.46)
SCHEMBL15173888 0.83 HCRTR1 (0.46)
SCHEMBL11896989 0.81 NPC1 (0.41) IL1BNPC1RAB9A
SCHEMBL15229464 0.81 IL1B (0.45) IL1BNPC1RAB9A
SCHEMBL2688541 0.81 NPC1 (0.41) IL1BNPC1RAB9A
SCHEMBL6523847 0.81 NPC1 (0.41) IL1BNPC1RAB9A
SCHEMBL13149783 0.80 IL1B (0.46) IL1BIDO1TDO2IRAK4CCNT1
SCHEMBL1598038 0.80 IDO1 (0.49) IL1BIDO1TDO2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020247445-A1 IMIDAZOLO DERIVATIVES, COMPOSITIONS AND METHODS AS OREXIN ANTAGONISTS HAGER BIOSCIENCES, LLC (US) 2020-12-10 WO disclosed
WO-2020247447-A1 PYRAZOLE AND IMIDAZOLE DERIVATIVES, COMPOSITIONS AND METHODS AS OREXIN ANTAGONISTS HAGER BIOSCIENCES, LLC (US) 2020-12-10 WO disclosed