SCHEMBL2276362

SCHEMBL2276362

COC(=O)c1ccc2c(C3CCCCC3)c3n(c2c1)C[C@@H](N(CCNC(=O)OC(C)(C)C)Cc1ccccc1)COc1ccccc1-3

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PRKCA P17252 1/20 0.56
MMP12 P39900 1/20 0.56
NR1I2 O75469 3/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
OPRM1 P35372 1/20 0.33
OPRK1 P41145 1/20 0.33
MDM2 Q00987 3/20 0.32
CNR2 P34972 2/20 0.32
NR1H4 Q96RI1 1/20 0.31
NPC1L1 Q9UHC9 3/20 0.31
BRD4 O60885 1/20 0.31
KDM4D Q6B0I6 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2276676 0.95 PRKCA (0.63) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL2276737 0.94 PRKCA (0.49) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL394842 0.90 PRKCA (0.65) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL2281023 0.89 PRKCA (0.55) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL392728 0.86 PRKCA (0.56) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL2279340 0.86 PRKCA (0.42) PRKCAMMP12CYP3A4CYP2C9OPRM1
SCHEMBL393735 0.85 PRKCA (0.75) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL2276740 0.84 PRKCA (0.49) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL4218773 0.83 PRKCA (0.44) PRKCAMMP12CYP3A4CYP2C9OPRM1
SCHEMBL393732 0.83 PRKCA (0.55) PRKCAMMP12NR1I2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7989438-B2 Therapeutic compounds ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2011-08-02 US disclosed