SCHEMBL22769992

SCHEMBL22769992

Fc1cc(Br)c(F)c(F)c1F.[MgH2]

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA7 P43166 1/20 0.33
CA13 Q8N1Q1 1/20 0.33
KDM1A O60341 2/20 0.31
KCNH2 Q12809 2/20 0.31
KDM1B Q8NB78 1/20 0.31
CES2 O00748 1/20 0.31
CES1 P23141 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1043011 0.97 CA12 (0.35) CA12CA1CA2CA7CA13
SCHEMBL31110619 0.81 CA1 (0.32) CA1CA2KDM1AKCNH2KDM1B
SCHEMBL4601309 0.77 CA12 (0.33) CA12CA1CA2CA7CA13
SCHEMBL21218726 0.77 AKR1B1 (0.34) KDM1AKCNH2KDM1B
SCHEMBL11884949 0.77 APEX1 (0.38) CA12CA1CA2CA7CA13
SCHEMBL7592418 0.74 SOS1 (0.38)
Bromide SCHEMBL8559956 0.74 CA1 (0.39) CA12CA1CA2CA7CA13
SCHEMBL7702552 0.73 CA1 (0.43) CA12CA1CA2CA7CA13
SCHEMBL41646 0.73 CA1 (0.43) CA12CA1CA2CA7CA13
SCHEMBL25200672 0.72 CYP3A4 (0.38) CA12CA1CA2CA7CA13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3750885-A1 COMPOUND HAVING BET INHIBITORY ACTIVITY AND PREPARATION METHOD AND USE THEREFOR Shanghai Haihe Pharmaceutical Co., Ltd. (CN) 2020-12-16 EP disclosed