SCHEMBL22779101

SCHEMBL22779101

C=C/C=C(\C)C#Cc1ccc(-c2ccnn2C)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP19A1 P11511 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
KCNH2 Q12809 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
PDE10A Q9Y233 1/20 0.35
PORCN Q9H237 1/20 0.34
SLC13A5 Q86YT5 1/20 0.34
CD274 Q9NZQ7 1/20 0.33
DRD1 P21728 1/20 0.33
PIK3CD O00329 1/20 0.33
PIK3CA P42336 1/20 0.33
PIK3CB P42338 1/20 0.33
PI4KA P42356 1/20 0.33
PIK3CG P48736 1/20 0.33
PI4KB Q9UBF8 1/20 0.33
ICMT O60725 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6852088 0.75 CYP1A2 (0.50) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL21258320 0.72 CYP1A2 (0.50) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL28561226 0.72 CYP1A2 (0.50) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL21258105 0.72 CYP1A2 (0.50) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL6852202 0.72 CYP1A2 (0.47) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL22779156 0.71 CYP1A2 (0.49) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL25011332 0.70 ACACB (0.44) CYP1A2PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL21258294 0.69 CYP1A2 (0.53) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL20001579 0.68 APP (0.44) CYP3A4ALDH1A1MAPT
SCHEMBL20216038 0.68 FFAR1 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3750881-A1 COMPOUND ACTING AS ANTIBIOTICS KBP Biosciences Co., Ltd. (CN) 2020-12-16 EP disclosed