SCHEMBL2279362

SCHEMBL2279362

COC(=O)c1ccc2c(C3CCCCC3)c3n(c2c1)C[C@H](OCC1CCCN1CCN(C)S(=O)(=O)NC(=O)OC(C)(C)C)COc1ccccc1-3

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PRKCA P17252 1/20 0.47
MMP12 P39900 1/20 0.47
NR1I2 O75469 8/20 0.37
KCNH2 Q12809 7/20 0.34
CYP3A4 P08684 3/20 0.34
SCN5A Q14524 2/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
SCN9A Q15858 4/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2276552 0.95 PRKCA (0.54) PRKCAMMP12NR1I2KCNH2CYP3A4
SCHEMBL2275224 0.90 PRKCA (0.49) PRKCAMMP12NR1I2KCNH2CYP3A4
SCHEMBL2279364 0.87 PRKCA (0.44) PRKCAMMP12NR1I2KCNH2CYP3A4
SCHEMBL2277316 0.87 PRKCA (0.34) PRKCAMMP12
SCHEMBL2277252 0.84 PRKCA (0.49) PRKCAMMP12NR1I2KCNH2CYP3A4
SCHEMBL4223402 0.84 PRKCA (0.57) PRKCAMMP12NR1I2KCNH2CYP3A4
SCHEMBL3685055 0.84 PRKCA (0.57) PRKCAMMP12NR1I2KCNH2CYP3A4
SCHEMBL4206442 0.84 PRKCA (0.37) PRKCAMMP12
SCHEMBL3685264 0.83 PRKCA (0.59) PRKCAMMP12NR1I2KCNH2CYP3A4
SCHEMBL2281723 0.83 PRKCA (0.59) PRKCAMMP12NR1I2KCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7989438-B2 Therapeutic compounds ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2011-08-02 US disclosed