SCHEMBL22804573

SCHEMBL22804573

COc1ccc(CNC2CC(=O)NC23CCC3)cc1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
TSHR P16473 3/20 0.46
LMNA P02545 1/20 0.46
SMN1; SMN2 Q16637 4/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 1/20 0.41
ALDH1A1 P00352 5/20 0.40
MAPT P10636 1/20 0.40
USP2 O75604 1/20 0.40
KDM1A O60341 1/20 0.40
GAA P10253 2/20 0.39
AKR1B1 P15121 1/20 0.38
BLM P54132 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
SSTR3 P32745 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29542941 0.81 MEN1 (0.45) MEN1KMT2ATSHRLMNASMN1; SMN2
SCHEMBL20041908 0.70 DDB1 (0.44) MEN1KMT2ATSHRSMN1; SMN2NPC1
SCHEMBL19559384 0.70 DDB1 (0.44) MEN1KMT2ATSHRSMN1; SMN2NPC1
SCHEMBL19559433 0.69 DDB1 (0.43) MEN1KMT2ATSHRSMN1; SMN2NPC1
SCHEMBL1350682 0.69 SMN1; SMN2 (0.47) MEN1KMT2ATSHRLMNASMN1; SMN2
SCHEMBL1350684 0.69 SMN1; SMN2 (0.47) MEN1KMT2ATSHRLMNASMN1; SMN2
SCHEMBL1350680 0.69 SMN1; SMN2 (0.47) MEN1KMT2ATSHRLMNASMN1; SMN2
SCHEMBL23126457 0.68 SMN1; SMN2 (0.47) MEN1KMT2ATSHRLMNASMN1; SMN2
SCHEMBL31681185 0.68 TSHR (0.47) MEN1KMT2ATSHRLMNASMN1; SMN2
SCHEMBL16914380 0.68 SMN1; SMN2 (0.47) MEN1KMT2ATSHRLMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3986886-A2 SUBSTITUTED PYRROLIDINE AMIDES V Grünenthal GmbH (DE) 2022-04-27 EP disclosed
WO-2020254552-A2 SUBSTITUTED PYRROLIDINE AMIDES V Grünenthal GmbH (DE) 2020-12-24 WO disclosed