SCHEMBL22809478

SCHEMBL22809478

CNCCOc1ccc2cc(OCC(F)(F)F)ccc2c1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.52
CYP17A1 P05093 2/20 0.52
CYP2C19 P33261 2/20 0.52
PDK2 Q15119 2/20 0.48
HTR1B P28222 2/20 0.47
HTR1D P28221 1/20 0.47
ALDH1A1 P00352 2/20 0.47
KDM4E B2RXH2 2/20 0.46
LMNA P02545 1/20 0.46
PPARG P37231 2/20 0.44
CYP1A2 P05177 1/20 0.42
CARM1 Q86X55 1/20 0.41
PRMT6 Q96LA8 1/20 0.41
CHRNB2 P17787 1/20 0.41
CHRNA4 P43681 1/20 0.41
GPR3 P46089 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22809479 0.78 CYP2C9 (0.53) CYP2C9CYP17A1CYP2C19PDK2ALDH1A1
SCHEMBL17303578 0.78 HTR1B (0.52) HTR1BHTR1DALDH1A1KDM4ELMNA
SCHEMBL19171717 0.77 HTR1B (0.47) PDK2HTR1BHTR1DALDH1A1KDM4E
Hydrochloric Acid SCHEMBL28351143 0.77 CYP2C9 (0.51) CYP2C9CYP17A1CYP2C19PDK2ALDH1A1
Hydrochloric Acid SCHEMBL30450085 0.77 CYP2C9 (0.51) CYP2C9CYP17A1CYP2C19PDK2ALDH1A1
SCHEMBL14431365 0.76 PDK2 (0.47) PDK2HTR1BHTR1DALDH1A1KDM4E
SCHEMBL5539798 0.76 HTR1B (0.58) CYP2C9CYP2C19HTR1BHTR1DALDH1A1
SCHEMBL10498275 0.75 CYP17A1 (0.57) CYP2C9CYP17A1CYP2C19ALDH1A1KDM4E
Hydrochloric Acid SCHEMBL27174649 0.75 HTR1B (0.56) CYP2C9CYP2C19HTR1BHTR1DALDH1A1
SCHEMBL1760893 0.74 L3MBTL1 (0.58) PDK2HTR1BHTR1DALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3487839-B1 AMIDE DERIVATIVES AS NAV1.7 AND NAV1.8 BLOCKERS RAQUALIA PHARMA INC (JP) 2020-12-23 EP disclosed