SCHEMBL22809643

SCHEMBL22809643

C=Cc1ccnc(NC(=O)C2CC2)n1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.45
RXFP1 Q9HBX9 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
ADORA2A P29274 2/20 0.43
ADORA3 P0DMS8 1/20 0.43
ADORA1 P30542 1/20 0.43
LMNA P02545 2/20 0.43
GSK3B P49841 7/20 0.43
ACVRL1 P37023 2/20 0.43
POLB P06746 1/20 0.43
ABL1 P00519 2/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
ADORA2B P29275 1/20 0.41
PIK3C3 Q8NEB9 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22809469 0.87 HPGD (0.46) HPGDRXFP1L3MBTL1ADORA2AADORA3
SCHEMBL30449743 0.77 GSK3B (0.56) HPGDRXFP1L3MBTL1ADORA2AADORA3
SCHEMBL29155745 0.77 POLB (0.64) HPGDRXFP1L3MBTL1ADORA2AADORA3
SCHEMBL2714790 0.76 KDM4E (0.61) HPGDRXFP1L3MBTL1ADORA2AADORA3
SCHEMBL11002946 0.73 HPGD (0.45) HPGDRXFP1L3MBTL1ADORA2AADORA3
SCHEMBL2715477 0.72 JAK1 (0.47) HPGDRXFP1L3MBTL1ADORA2AADORA3
SCHEMBL4550418 0.71 ADORA1 (0.45) HPGDRXFP1L3MBTL1ADORA2AADORA3
SCHEMBL22186405 0.71 KDM4E (0.58) HPGDRXFP1L3MBTL1ADORA2AADORA3
SCHEMBL4710625 0.70 HPGD (0.47) HPGDADORA2AADORA3ADORA1LMNA
SCHEMBL4710626 0.70 HPGD (0.47) HPGDADORA2AADORA3ADORA1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3487839-B1 AMIDE DERIVATIVES AS NAV1.7 AND NAV1.8 BLOCKERS RAQUALIA PHARMA INC (JP) 2020-12-23 EP disclosed