SCHEMBL4550418

SCHEMBL4550418

O=C(Nc1nccc(C(O)=C2CC2)n1)C1CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 5/20 0.45
ADORA2A P29274 4/20 0.45
ADORA3 P0DMS8 2/20 0.45
LMNA P02545 1/20 0.44
KDM4E B2RXH2 1/20 0.44
KDM5A P29375 1/20 0.44
JMJD1C Q15652 1/20 0.44
KDM3A Q9Y4C1 1/20 0.44
ACVRL1 P37023 2/20 0.43
HPGD P15428 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
GSK3B P49841 4/20 0.41
POLB P06746 1/20 0.41
ABL1 P00519 1/20 0.40
JAK1 P23458 1/20 0.39
TYK2 P29597 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
ADORA2B P29275 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2714790 0.85 KDM4E (0.61) ADORA1ADORA2AADORA3LMNAKDM4E
SCHEMBL30449743 0.84 GSK3B (0.56) ADORA1ADORA2AADORA3LMNAKDM4E
SCHEMBL22186405 0.80 KDM4E (0.58) ADORA1ADORA2AADORA3LMNAKDM4E
SCHEMBL2715477 0.79 JAK1 (0.47) ADORA1ADORA2AADORA3LMNAKDM4E
SCHEMBL4550822 0.77 ADORA1 (0.47) ADORA1ADORA2AADORA3KDM4EHPGD
SCHEMBL29155745 0.75 POLB (0.64) ADORA1ADORA2AADORA3LMNAKDM4E
SCHEMBL22809469 0.72 HPGD (0.46) ADORA1ADORA2AADORA3LMNAACVRL1
SCHEMBL18906054 0.72 ADORA1 (0.50) ADORA1ADORA2AADORA3LMNAKDM4E
SCHEMBL22809643 0.71 HPGD (0.45) ADORA1ADORA2AADORA3LMNAACVRL1
SCHEMBL18266119 0.71 KDM4E (0.58) ADORA1ADORA2AADORA3LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012053186-A1 ARYLAMIDE DERIVATIVES AS TTX-S BLOCKERS RAQUALIA PHARMA INC. (JP) 2012-04-26 WO disclosed