SCHEMBL22809648

SCHEMBL22809648

Cc1cc(C(=O)O)nc(NC(=O)C2CCC2)n1

nearest known ligand 0.53

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 7/20 0.53
ADORA2A P29274 4/20 0.50
ADORA3 P0DMS8 3/20 0.50
RAB9A P51151 2/20 0.46
NPSR1 Q6W5P4 3/20 0.44
LMNA P02545 1/20 0.44
ATAD2 Q6PL18 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
NPC1 O15118 1/20 0.40
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2713671 0.94 ADORA1 (0.51) ADORA1ADORA2AADORA3RAB9ANPSR1
SCHEMBL30450912 0.81 ADORA1 (0.47) ADORA1ADORA2AADORA3RAB9ANPSR1
SCHEMBL4550822 0.81 ADORA1 (0.47) ADORA1ADORA2AADORA3RAB9ANPSR1
SCHEMBL18266209 0.80 MAPT (0.39) ADORA1ADORA2AADORA3RAB9ANPSR1
SCHEMBL2713731 0.80 HSD17B10 (0.49) ADORA1ADORA2AADORA3RAB9ANPSR1
SCHEMBL18266606 0.79 MAPT (0.38) ADORA1ADORA2AADORA3RAB9ANPSR1
SCHEMBL2713871 0.77 CYP1A2 (0.58) ADORA1ADORA3RAB9ALMNASMN1; SMN2
SCHEMBL1178837 0.76 MCHR1 (0.45) KDM4E
SCHEMBL22186405 0.75 KDM4E (0.58) ADORA1ADORA2AADORA3RAB9ALMNA
SCHEMBL18266404 0.75 ADORA1 (0.47) ADORA1ADORA2AADORA3RAB9ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3487839-B1 AMIDE DERIVATIVES AS NAV1.7 AND NAV1.8 BLOCKERS RAQUALIA PHARMA INC (JP) 2020-12-23 EP disclosed