SCHEMBL4550822

SCHEMBL4550822

Cc1cc(C(O)=C2CC2)nc(NC(=O)C2CC2)n1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 5/20 0.47
ADORA2A P29274 3/20 0.47
ADORA3 P0DMS8 2/20 0.47
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 1/20 0.41
NPSR1 Q6W5P4 1/20 0.39
HPGD P15428 1/20 0.39
RAB9A P51151 2/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
NPC1 O15118 1/20 0.39
VCP P55072 2/20 0.38
POLB P06746 1/20 0.38
AHR P35869 1/20 0.37
MAPT P10636 1/20 0.37
ABL1 P00519 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2713671 0.86 ADORA1 (0.51) ADORA1ADORA2AADORA3ALDH1A1KDM4E
SCHEMBL30450912 0.82 ADORA1 (0.47) ADORA1ADORA2AADORA3ALDH1A1KDM4E
SCHEMBL2713731 0.81 HSD17B10 (0.49) ADORA1ADORA2AADORA3ALDH1A1KDM4E
SCHEMBL22809648 0.81 ADORA1 (0.53) ADORA1ADORA2AADORA3ALDH1A1KDM4E
SCHEMBL4550418 0.77 ADORA1 (0.45) ADORA1ADORA2AADORA3KDM4EHPGD
SCHEMBL18266404 0.73 ADORA1 (0.47) ADORA1ADORA2AADORA3ALDH1A1KDM4E
SCHEMBL18266209 0.72 MAPT (0.39) ADORA1ADORA2AADORA3KDM4ENPSR1
SCHEMBL15358619 0.71 ADORA1 (0.45) ADORA1ADORA2AADORA3ALDH1A1KDM4E
SCHEMBL18266606 0.71 MAPT (0.38) ADORA1ADORA2AADORA3KDM4ENPSR1
Hydrochloric Acid SCHEMBL15350578 0.70 ADORA1 (0.44) ADORA1ADORA2AADORA3ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012053186-A1 ARYLAMIDE DERIVATIVES AS TTX-S BLOCKERS RAQUALIA PHARMA INC. (JP) 2012-04-26 WO disclosed