SCHEMBL22822296

SCHEMBL22822296

CCOC(=O)C1(NC(=O)N[C@]2(C)CC[C@]3(C)CC[C@]4(C)C5=CC=C6C(=CC(=O)C(O)=C6C)[C@]5(C)CC[C@@]4(C)[C@@H]3C2)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PRDX1 Q06830 16/20 1.00
NR4A1 P22736 2/20 0.75
TERT O14746 1/20 0.75
PTPN1 P18031 1/20 0.67
CASP1 P29466 1/20 0.67
ABHD6 Q9BV23 1/20 0.67
KDM4E B2RXH2 1/20 0.67
TP53 P04637 1/20 0.67
CYP3A4 P08684 1/20 0.67
MAPT P10636 1/20 0.67
HPGD P15428 1/20 0.67
ALOX15 P16050 1/20 0.67
ALOX12 P18054 1/20 0.67
MAPK1 P28482 1/20 0.67
SMN1; SMN2 Q16637 1/20 0.67
TDP1 Q9NUW8 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18781890 0.89 PRDX1 (0.80) PRDX1NR4A1TERTPTPN1CASP1
SCHEMBL18781883 0.88 PRDX1 (0.83) PRDX1NR4A1
SCHEMBL22822210 0.87 PRDX1 (1.00) PRDX1NR4A1PTPN1CASP1ABHD6
SCHEMBL22822453 0.87 PRDX1 (1.00) PRDX1NR4A1PTPN1CASP1ABHD6
SCHEMBL18781882 0.86 PRDX1 (0.76) PRDX1NR4A1TERTPTPN1CASP1
SCHEMBL12395123 0.86 NR4A1 (1.00) PRDX1NR4A1TERTPTPN1CASP1
SCHEMBL22822454 0.84 PRDX1 (1.00) PRDX1NR4A1PTPN1CASP1ABHD6
SCHEMBL22822305 0.84 PRDX1 (1.00) PRDX1
SCHEMBL22822306 0.82 PRDX1 (1.00) PRDX1TERT
SCHEMBL25512294 0.81 NR4A1 (0.73) PRDX1NR4A1TERTPTPN1CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020253814-A1 TRIPTERINE DERIVATIVES, PREPARATION METHOD THEREFOR AND USE THEREOF 中国科学院上海药物研究所 2020-12-24 WO disclosed