SCHEMBL22825554

SCHEMBL22825554

CCCCCCOc1ccc(-c2cc(C(F)(F)F)nn2C)c(O)c1-c1cncc(C=N)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SPHK2 Q9NRA0 3/20 0.35
THRA P10827 1/20 0.32
THRB P10828 1/20 0.32
STIM1 Q13586 2/20 0.31
ORAI1 Q96D31 2/20 0.31
SCN9A Q15858 1/20 0.31
ALOX5 P09917 1/20 0.31
PTGS1 P23219 1/20 0.31
PTGS2 P35354 1/20 0.31
S1PR1 P21453 2/20 0.30
S1PR4 O95977 1/20 0.30
S1PR5 Q9H228 1/20 0.30
HDAC3 O15379 1/20 0.30
HDAC4 P56524 1/20 0.30
HDAC1 Q13547 1/20 0.30
HDAC7 Q8WUI4 1/20 0.30
HDAC2 Q92769 1/20 0.30
HDAC10 Q969S8 1/20 0.30
HDAC11 Q96DB2 1/20 0.30
HDAC8 Q9BY41 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22825391 0.97 SCN9A (0.33) SPHK2STIM1ORAI1SCN9AALOX5
SCHEMBL21786426 0.89 PPARD (0.33) THRATHRBSTIM1ORAI1S1PR1
SCHEMBL21786487 0.86 USP7 (0.36) SCN9A
SCHEMBL22791224 0.85 PPARD (0.34) STIM1ORAI1SCN9A
SCHEMBL22825614 0.84 STIM1 (0.35) STIM1ORAI1SCN9APTGS1PTGS2
SCHEMBL21786433 0.82 SCN9A (0.37) SCN9A
SCHEMBL24127463 0.81 AGER (0.32) SPHK2
SCHEMBL21786504 0.80 PTGDR2 (0.36) STIM1ORAI1SCN9AALOX5PTGS1
SCHEMBL21786492 0.77 DYRK3 (0.32) STIM1ORAI1ALOX5PTGS1PTGS2
SCHEMBL22790953 0.75 PPARD (0.34) STIM1ORAI1SCN9APTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020257261-A1 SUBSTITUTED HETEROCYCLES AS c-MYC TARGETING AGENTS NORTHWESTERN UNIVERSITY (US) 2020-12-24 WO disclosed