SCHEMBL2283178

SCHEMBL2283178

CN1CCN(Cc2ccc(-c3cc4nccc(Oc5ccc(N)cc5F)c4s3)cc2)CC1

nearest known ligand 0.63

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MET P08581 11/20 0.63
KDR P35968 10/20 0.63
SRC P12931 6/20 0.49
MST1R Q04912 1/20 0.47
ABL1 P00519 1/20 0.45
ABL2 P42684 1/20 0.45
AXL P30530 1/20 0.42
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL306763 0.92 MET (0.54) METKDRSRCMST1RAXL
SCHEMBL13166733 0.90 KDR (0.52) METKDRSRCMST1RAXL
SCHEMBL306277 0.89 MST1R (0.58) METKDRSRCMST1RABL1
SCHEMBL10223932 0.88 MET (0.65) METKDRSRCMST1RAXL
SCHEMBL3617148 0.88 MET (0.60) METKDRMST1R
SCHEMBL13169019 0.88 MET (0.67) METKDRSRCMST1RABL1
SCHEMBL13167210 0.86 MET (0.56) METKDRMST1R
SCHEMBL13167395 0.84 MET (0.69) METKDRMST1R
SCHEMBL10223924 0.84 MET (0.48) METKDRMST1R
SCHEMBL14136730 0.84 MET (0.77) METKDRMST1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8003662-B2 Heterobicyclic thiophene compounds and methods of use ARRAY BIOPHARMA, INC. (US) 2011-08-23 US disclosed
EP-1989211-A2 HETEROBICYCLIC THIOPHENE COMPOUNDS FOR THE TREATMENT OF CANCER Array Biopharma, Inc. (US) 2008-11-12 EP disclosed
WO-2008063202-A2 HETEROBICYCLIC THIOPHENE COMPOUNDS FOR THE TREATMENT OF CANCER ARRAY BIOPHARMA INC. (US) 2008-05-29 WO disclosed
US-20070197537-A1 Heterobicyclic thiophene compounds and methods of use ARRAY BIOPHARMA, INC. 2007-08-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070197537-A1 Heterobicyclic thiophene compounds and methods of use ERBB2, LCK, SRC MET 142/4885KDR 419/4885SRC 3/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.