SCHEMBL2283665

SCHEMBL2283665

Cc1cc(C)cc(CC(N[S+]([O-])C(C)(C)C)c2cccnc2)c1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.38
CYP2D6 P10635 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
MAPT P10636 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.33
MAPK1 P28482 1/20 0.33
KCNA5 P22460 1/20 0.32
THRB P10828 1/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
SLC6A3 Q01959 1/20 0.32
TDP1 Q9NUW8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21259925 0.81 KCNN4 (0.38) LMNAKCNA5SLC6A2SLC6A4SLC6A3
SCHEMBL2289154 0.76
SCHEMBL28643199 0.76 KDM4E (0.33) CYP3A4CYP2D6CYP1A2CYP2C9CYP2C19
SCHEMBL29571827 0.76 KDM4E (0.33) CYP3A4CYP2D6CYP1A2CYP2C9CYP2C19
SCHEMBL28643197 0.76 KDM4E (0.33) CYP3A4CYP2D6CYP1A2CYP2C9CYP2C19
SCHEMBL24931445 0.76 KDM4E (0.33) CYP3A4CYP2D6CYP1A2CYP2C9CYP2C19
SCHEMBL28921258 0.76 KDM4E (0.33) CYP3A4CYP2D6CYP1A2CYP2C9CYP2C19
SCHEMBL24968597 0.76 KDM4E (0.33) CYP3A4CYP2D6CYP1A2CYP2C9CYP2C19
SCHEMBL28921359 0.76 KDM4E (0.33) CYP3A4CYP2D6CYP1A2CYP2C9CYP2C19
SCHEMBL29571429 0.76 KDM4E (0.33) CYP3A4CYP2D6CYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7989394-B2 Substituted 1-(azolin-2-yl)-amino-2-aryl-1-hetaryl-ethane compounds BASF SE (DE) 2011-08-02 US disclosed