SCHEMBL22840481

SCHEMBL22840481

O=Cc1c(O)ccc2[nH]c(C(=O)NCCNCCO)cc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.43
ALDH1A1 P00352 3/20 0.43
HPGD P15428 2/20 0.43
TP53 P04637 1/20 0.41
CASP1 P29466 1/20 0.41
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
AKR1C3 P42330 1/20 0.39
HSD17B10 Q99714 1/20 0.39
MAPT P10636 1/20 0.38
NPC1 O15118 1/20 0.37
POLB P06746 1/20 0.37
RAB9A P51151 1/20 0.37
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
DRD2 P14416 2/20 0.36
HTR1A P08908 1/20 0.36
HTR2A P28223 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30406065 0.83 NPC1 (0.44) KDM4EALDH1A1HPGDCA12CA1
SCHEMBL2562212 0.83 NPC1 (0.44) KDM4EALDH1A1HPGDCA12CA1
SCHEMBL2567378 0.83 ALOX15 (0.47) KDM4EALDH1A1CA12CA1CA2
SCHEMBL30406074 0.82 HTR2C (0.55) KDM4EALDH1A1HPGDCA12CA1
SCHEMBL2565847 0.82 HTR2C (0.55) KDM4EALDH1A1HPGDCA12CA1
SCHEMBL14916752 0.77 KDM4E (0.60) KDM4EALDH1A1HPGDHSD17B10MAPT
SCHEMBL22840478 0.77 HRH4 (0.42) KDM4EALDH1A1HPGDCA12CA1
SCHEMBL30406446 0.77 KDM4E (0.60) KDM4EALDH1A1HPGDHSD17B10MAPT
SCHEMBL14925523 0.75 KDM4E (0.50) KDM4EALDH1A1HPGDHSD17B10MAPT
SCHEMBL7471060 0.73 KDM4E (0.52) KDM4EALDH1A1HPGDHSD17B10MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3799870-A1 IRE-1A INHIBITORS Fosun Orinove Pharmatech, Inc. (CN) 2021-04-07 EP disclosed
EP-3409276-B1 IRE-1A INHIBITORS FOSUN ORINOVE PHARMATECH INC (CN) 2020-12-30 EP disclosed