SCHEMBL2284198

SCHEMBL2284198

NC(=O)c1c(O)c2ccccc2oc1=O

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.71
CA9 Q16790 1/20 0.71
LMNA P02545 5/20 0.61
HPGD P15428 1/20 0.61
ALDH1A1 P00352 4/20 0.60
KDM4E B2RXH2 3/20 0.60
SMN1; SMN2 Q16637 3/20 0.60
MAPT P10636 1/20 0.60
HTT P42858 4/20 0.58
NQO1 P15559 4/20 0.56
TP53 P04637 3/20 0.56
MEN1 O00255 2/20 0.56
KMT2A Q03164 2/20 0.56
TSHR P16473 2/20 0.56
MAPK1 P28482 2/20 0.56
ABCB11 O95342 1/20 0.56
CYP1A2 P05177 1/20 0.56
CYP3A4 P08684 1/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2C19 P33261 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29901650 0.84 CA12 (0.73) CA12CA9LMNAHPGDALDH1A1
SCHEMBL1648027 0.84 CA12 (0.73) CA12CA9LMNAHPGDALDH1A1
SCHEMBL3527681 0.83 CA12 (1.00) CA12CA9LMNAHPGDALDH1A1
SCHEMBL30933370 0.83 CA12 (1.00) CA12CA9LMNAHPGDALDH1A1
SCHEMBL10613511 0.81 CA12 (0.69) CA12CA9LMNAHPGDALDH1A1
SCHEMBL1850238 0.81 ALDH1A1 (0.56) CA12CA9LMNAHPGDALDH1A1
SCHEMBL9278433 0.80 NQO1 (0.58) CA12CA9LMNAHPGDALDH1A1
SCHEMBL29801774 0.80 ALDH1A1 (0.51) CA12CA9LMNAHPGDALDH1A1
SCHEMBL24864745 0.79 CA12 (0.65) CA12CA9LMNAHPGDALDH1A1
SCHEMBL17169389 0.79 CA12 (0.69) CA12CA9LMNAHPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 41 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0550493-A1 ANTHELMINTIC AND ANTICOCCIDAL 3-CARBAMOYL-4-HYDROXYCOUMARINS, METHOD OF USE AND COMPOSITIONS. UPJOHN CO (US) 1993-07-14 EP claimed
WO-1992006083-A1 ANTHELMINTIC AND ANTICOCCIDAL 3-CARBAMOYL-4-HYDROXYCOUMARINS, METHOD OF USE AND COMPOSITIONS THE UPJOHN COMPANY (US) 1992-04-16 WO claimed
US-4766144-A 3-carbamoyl-4-hydroxy-coumarins for combating parasitic heiminths BAYER AKTIENGESELLSCHAFT (DE) 1988-08-23 US claimed
EP-0241834-A2 Use of 3-carbamoyl-4-hydroxy-cumarines in combating parasiticidal helminths, 3-carbamoyl-4-hydroxy-cumarines and their preparation BAYER AG (DE) 1987-10-21 EP claimed
EP-0038427-A1 3-Carbamoyl-4-hydroxy-cumarines, process for their preparation and their use as pesticides BAYER AG (DE) 1981-10-28 EP claimed
EP-2295053-B1 Novel 2H-chromen-2-one-3-carboxamides for medical uses INST MATERIA MEDICA CAMS (CN) 2016-10-19 EP disclosed
US-20110263642-A1 METHODS FOR TREATMENT OF MULTIPLE SCLEROSIS FIBROGEN, INC. (US) 2011-10-27 US disclosed
EP-2341904-A1 METHODS FOR TREATMENT OF MULTIPLE SCLEROSIS Fibrogen, Inc. (US) 2011-07-13 EP disclosed
WO-2010024908-A1 METHODS FOR TREATMENT OF MULTIPLE SCLEROSIS FIBROGEN, INC. (US) 2010-03-04 WO disclosed
EP-1664332-A4 KINASE AND PHOSPHATASE ASSAYS INVITROGEN CORP (US) 2008-05-14 EP disclosed
WO-2008054695-A2 COMPOSITION AND METHOD FOR ETIOLOGICAL TREATMENT AND PREVENTION OF DISEASES AND/OR COMPLICATIONS ASSOCIATED WITH CHRONIC GLUCOSE METABOLISM DESTABILIZATION GUFFEY MANNING V (US) 2008-05-08 WO disclosed
US-20080102137-A1 Composition and method for etiological treatment and prevention of diseases and/or complications associated with chronic glucose metabolism destabilization GUFFEY MANNING V R 2008-05-01 US disclosed
EP-0241834-A3 USE OF 3-CARBAMOYL-4-HYDROXY-CUMARINES IN COMBATING PARASITICIDAL HELMINTHS, 3-CARBAMOYL-4-HYDROXY-CUMARINES AND THEIR PREPARATION BAYER AG (DE) 1988-10-26 EP disclosed
US-4766144-A 3-carbamoyl-4-hydroxy-coumarins for combating parasitic heiminths BAYER AKTIENGESELLSCHAFT (DE) 1988-08-23 US disclosed
US-4766144-A 3-carbamoyl-4-hydroxy-coumarins for combating parasitic heiminths BAYER AKTIENGESELLSCHAFT (DE) 1988-08-23 US disclosed
EP-0241834-A2 Use of 3-carbamoyl-4-hydroxy-cumarines in combating parasiticidal helminths, 3-carbamoyl-4-hydroxy-cumarines and their preparation BAYER AG (DE) 1987-10-21 EP disclosed
EP-0241834-A2 Use of 3-carbamoyl-4-hydroxy-cumarines in combating parasiticidal helminths, 3-carbamoyl-4-hydroxy-cumarines and their preparation BAYER AG (DE) 1987-10-21 EP disclosed
EP-0038427-A1 3-Carbamoyl-4-hydroxy-cumarines, process for their preparation and their use as pesticides BAYER AG (DE) 1981-10-28 EP disclosed
EP-0038427-A1 3-Carbamoyl-4-hydroxy-cumarines, process for their preparation and their use as pesticides BAYER AG (DE) 1981-10-28 EP disclosed
EP-0038427-A1 3-Carbamoyl-4-hydroxy-cumarines, process for their preparation and their use as pesticides BAYER AG (DE) 1981-10-28 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110263642-A1 METHODS FOR TREATMENT OF MULTIPLE SCLEROSIS PMP22, MAG, NEFM CA12 821/4885CA9 2529/4885LMNA 2864/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.