SCHEMBL22860146

SCHEMBL22860146

CSc1ncc(CO)c(Nc2c(F)cccc2F)n1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.51
MAPK1 P28482 1/20 0.41
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CDK9 P50750 2/20 0.38
CCNT1 O60563 1/20 0.38
SYK P43405 3/20 0.36
CCNA2 P20248 1/20 0.36
CDK2 P24941 1/20 0.36
CCNA1 P78396 1/20 0.36
PIM1 P11309 2/20 0.35
BAD Q92934 2/20 0.35
PIM2 Q9P1W9 2/20 0.35
RXFP1 Q9HBX9 1/20 0.35
JAK1 P23458 3/20 0.35
TYK2 P29597 3/20 0.35
JAK3 P52333 3/20 0.35
JAK2 O60674 1/20 0.35
MERTK Q12866 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6344153 0.80 HTT (0.46) HTTMAPK1MAPTSYKCCNA2
SCHEMBL4712352 0.80 HTT (0.51) HTTMAPK1ALDH1A1MAPTSMN1; SMN2
SCHEMBL4846993 0.77 MAPK1 (0.39) HTTMAPK1ALDH1A1MAPTSMN1; SMN2
SCHEMBL28039439 0.77 HTT (0.52) HTTMAPK1ALDH1A1MAPTSMN1; SMN2
SCHEMBL26107898 0.75 HTT (0.47) HTTMAPK1CDK9SYKCCNA2
SCHEMBL30596936 0.75 HTT (0.47) HTTMAPK1CDK9SYKCCNA2
SCHEMBL6619405 0.75 HTT (0.42) HTTMAPK1ALDH1A1MAPTSMN1; SMN2
SCHEMBL1521589 0.75 HTT (0.51) HTTMAPK1ALDH1A1MAPTSMN1; SMN2
SCHEMBL4854253 0.75 HTT (0.72) HTTMAPK1ALDH1A1MAPTSMN1; SMN2
SCHEMBL6617756 0.74 HTT (0.54) HTTMAPK1SYKPIM1JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3993802-A1 HETEROCYCLIC COMPOUNDS AS KINASE INHIBITORS Nuvation Bio Inc. (US) 2022-05-11 EP disclosed
CN-114340634-A Heterocyclic compounds as kinase inhibitors 诺维逊生物股份有限公司 2022-04-12 CN disclosed
WO-2021003314-A1 HETEROCYCLIC COMPOUNDS AS KINASE INHIBITORS NUVATION BIO INC. (US) 2021-01-07 WO disclosed