SCHEMBL22866407

SCHEMBL22866407

Cc1nc2c(Cl)ncc(C#N)c2c(=O)[nH]1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 7/20 0.39
MAPK1 P28482 1/20 0.38
GAA P10253 1/20 0.37
TYMS P04818 2/20 0.36
IDH1 O75874 4/20 0.35
CSNK1A1 P48729 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34
PIM1 P11309 1/20 0.34
PIM2 Q9P1W9 1/20 0.34
CDK4 P11802 1/20 0.33
CCND1 P24385 1/20 0.33
ALDH1A1 P00352 1/20 0.33
KDM4E B2RXH2 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29561211 1.00 PARP1 (0.39) PARP1MAPK1GAATYMSIDH1
SCHEMBL22866409 0.85 MAPK1 (0.39) PARP1MAPK1GAATYMSALDH1A1
SCHEMBL29559852 0.85 MAPK1 (0.39) PARP1MAPK1GAATYMSALDH1A1
SCHEMBL22866406 0.78 PARP1 (0.42) PARP1MAPK1TYMSPIM1PIM2
SCHEMBL29559956 0.78 PARP1 (0.42) PARP1MAPK1TYMSPIM1PIM2
SCHEMBL22866745 0.75 PARP1 (0.47) PARP1GAATYMSALDH1A1KDM4E
SCHEMBL29559925 0.75 PARP1 (0.47) PARP1GAATYMSALDH1A1KDM4E
SCHEMBL23900415 0.71 MAPK1 (0.56) MAPK1GAAIDH1ALDH1A1KDM4E
SCHEMBL22866432 0.71 GAA (0.45) PARP1MAPK1GAATYMSPIM1
SCHEMBL29559893 0.71 GAA (0.45) PARP1MAPK1GAATYMSPIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021003157-A1 EIF4E-INHIBITING 4-OXO-3,4-DIHYDROPYRIDO[3,4-D]PYRIMIDINE COMPOUNDS EFFECTOR THERAPEUTICS, INC. (US) 2021-01-07 WO disclosed