SCHEMBL22868067

SCHEMBL22868067

Cc1ccc2c(c1)C(N)CS2

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.35
SMN1; SMN2 Q16637 4/20 0.35
MAPT P10636 1/20 0.35
AADAT Q8N5Z0 2/20 0.35
CHRNB2 P17787 1/20 0.34
CHRNA4 P43681 1/20 0.34
NPSR1 Q6W5P4 2/20 0.33
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33
HPGD P15428 2/20 0.33
ALOX15 P16050 2/20 0.33
ALDH1A1 P00352 2/20 0.33
MEN1 O00255 1/20 0.33
ALOX12 P18054 1/20 0.33
BRCA1 P38398 1/20 0.33
KMT2A Q03164 1/20 0.33
HSD17B10 Q99714 1/20 0.33
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7914321 0.78 CA1 (0.38) KDM4ESMN1; SMN2MAPTCHRNB2CHRNA4
SCHEMBL10183439 0.77 KDM4E (0.38) KDM4ESMN1; SMN2MAPTCHRNB2CHRNA4
SCHEMBL8144693 0.71 HTR2A (0.41) MAPTHPGDALDH1A1MEN1ALOX12
SCHEMBL8520772 0.69 EPHX2 (0.55) KDM4ESMN1; SMN2MAPTAADATNPSR1
SCHEMBL9835145 0.68 RCE1 (0.47) SMN1; SMN2MAPTLMNAHTTHPGD
SCHEMBL12253322 0.67 NOS3 (0.34) AADATCHRNB2CHRNA4HPGDALOX15
SCHEMBL464509 0.67 EPHX2 (0.37) KDM4ESMN1; SMN2MAPTCHRNB2CHRNA4
SCHEMBL464506 0.65 EPHX2 (0.36) KDM4ESMN1; SMN2MAPTCHRNB2CHRNA4
SCHEMBL31705254 0.65 KDM1A (0.41) HTR2CSLC6A2
SCHEMBL18325979 0.64 CYP2A6 (0.36) SMN1; SMN2CHRNB2CHRNA4HPGDALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021003295-A1 MODULATORS OF HSD17B13 AND METHODS OF USE THEREOF REGENERON PHARMACEUTICALS, INC. (US) 2021-01-07 WO disclosed