SCHEMBL2288030

SCHEMBL2288030

CN1CCC(C(=O)Nc2ccc(Oc3ccnc4cc(I)sc34)c(F)c2)C1=O

nearest known ligand 0.62

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MET P08581 20/20 0.62
KDR P35968 16/20 0.62
MST1R Q04912 1/20 0.47
AXL P30530 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2284731 0.84 MET (0.61) METKDRMST1R
SCHEMBL2281890 0.84 MET (0.51) METKDR
SCHEMBL3621621 0.79 MET (0.55) METKDR
SCHEMBL2538072 0.79 MET (0.53) METKDR
SCHEMBL3109405 0.78 MET (0.56) METKDRAXL
SCHEMBL895182 0.77 MET (1.00) METKDRMST1R
SCHEMBL896308 0.77 MET (0.90) METKDRMST1R
SCHEMBL12410932 0.76 MET (0.63) METKDRMST1RAXL
SCHEMBL895880 0.76 MET (0.86) METKDRMST1R
SCHEMBL13167191 0.76 MET (0.49) METKDRMST1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8003662-B2 Heterobicyclic thiophene compounds and methods of use ARRAY BIOPHARMA, INC. (US) 2011-08-23 US disclosed
US-20070197537-A1 Heterobicyclic thiophene compounds and methods of use ARRAY BIOPHARMA, INC. 2007-08-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070197537-A1 Heterobicyclic thiophene compounds and methods of use ERBB2, LCK, SRC MET 142/4885KDR 419/4885MST1R 656/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.