SCHEMBL22890819

SCHEMBL22890819

COC(=O)c1nc(C2CC2)c(C#N)c(C)c1C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 5/20 0.48
GAA P10253 6/20 0.43
ALDH1A1 P00352 5/20 0.43
HPGD P15428 5/20 0.43
KDM4E B2RXH2 3/20 0.42
PKM P14618 1/20 0.41
NPSR1 Q6W5P4 1/20 0.38
CASP1 P29466 2/20 0.36
CASP7 P55210 2/20 0.36
HSD17B10 Q99714 2/20 0.36
MAPK10 P53779 1/20 0.36
TSHR P16473 2/20 0.34
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
IDH1 O75874 2/20 0.34
MAPT P10636 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22890502 0.84 LRRK2 (0.48) LRRK2GAAKDM4EPKMHSD17B10
SCHEMBL21847824 0.80 NPSR1 (0.52) LRRK2GAAALDH1A1HPGDKDM4E
SCHEMBL29496233 0.80 NPSR1 (0.52) LRRK2GAAALDH1A1HPGDKDM4E
SCHEMBL22890816 0.76 ALDH1A1 (0.47) LRRK2GAAALDH1A1HPGDKDM4E
SCHEMBL22890865 0.74 ALDH1A1 (0.44) LRRK2GAAALDH1A1HPGDKDM4E
SCHEMBL22890872 0.72 LRRK2 (0.44) LRRK2GAAALDH1A1HPGDKDM4E
SCHEMBL22890764 0.72 ALDH1A1 (0.43) LRRK2GAAALDH1A1HPGDKDM4E
SCHEMBL22890405 0.72 ALDH1A1 (0.43) LRRK2GAAALDH1A1HPGDKDM4E
SCHEMBL21847851 0.72 ALDH1A1 (0.56) LRRK2GAAALDH1A1HPGDKDM4E
SCHEMBL29496196 0.72 ALDH1A1 (0.56) LRRK2GAAALDH1A1HPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021007477-A1 INDAZOLES AND AZAINDAZOLES AS LRRK2 INHIBITORS E-SCAPE BIO, INC. (US) 2021-01-14 WO disclosed