SCHEMBL22904233

SCHEMBL22904233

O=C1Cc2cnc(Br)cc2C(=O)N1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TDP2 O95551 19/20 0.51
CASP3 P42574 1/20 0.44
CASP7 P55210 1/20 0.44
CASP9 P55211 1/20 0.44
CASP6 P55212 1/20 0.44
CASP8 Q14790 1/20 0.44
MAP3K14 Q99558 1/20 0.44
CMA1 P23946 1/20 0.39
AHR P35869 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30780152 1.00 TDP2 (0.51) TDP2CASP3CASP7CASP9CASP6
SCHEMBL30099759 0.75 CA12 (0.41)
SCHEMBL25300707 0.75 AHR (0.49) TDP2CMA1AHR
SCHEMBL6530104 0.72 PDE3B (0.44) TDP2CMA1AHR
SCHEMBL23092822 0.72 TDP2 (0.47) TDP2CASP3CASP7CASP9CASP6
SCHEMBL29861982 0.72 TDP2 (0.47) TDP2CASP3CASP7CASP9CASP6
SCHEMBL30015036 0.71 TDP2 (0.80) TDP2CASP3CASP7CASP9CASP6
SCHEMBL22904167 0.71 TDP2 (0.80) TDP2CASP3CASP7CASP9CASP6
SCHEMBL22885217 0.69 TDP2 (0.51) TDP2CASP3CASP7CASP9CASP6
SCHEMBL30699001 0.69 TDP2 (0.51) TDP2CASP3CASP7CASP9CASP6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4577546-A1 NAPHTHYRIDINE COMPOUNDS FOR INHIBITION OF RAF KINASES Enliven Inc. (US) 2025-07-02 EP disclosed
WO-2024044713-A1 NAPHTHYRIDINE COMPOUNDS FOR INHIBITION OF RAF KINASES ENLIVEN INC. (US) 2024-02-29 WO disclosed
WO-2024044713-A1 NAPHTHYRIDINE COMPOUNDS FOR INHIBITION OF RAF KINASES ENLIVEN INC. (US) 2024-02-29 WO disclosed
WO-2021011631-A1 FUSED-GLUTARIMIDE CRBN LIGANDS AND USES THEREOF KYMERA THERAPEUTICS, INC. (US) 2021-01-21 WO disclosed