SCHEMBL22905342

SCHEMBL22905342

CNCCc1ccc2c(c1)OC(F)(F)O2

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.46
TP53 P04637 1/20 0.46
CYP1A2 P05177 1/20 0.46
ALOX15 P16050 1/20 0.46
TSHR P16473 1/20 0.46
NFKB1 P19838 1/20 0.46
MAPK1 P28482 1/20 0.46
THPO P40225 1/20 0.46
HIF1A Q16665 1/20 0.46
HSD17B10 Q99714 1/20 0.46
TAAR1 Q96RJ0 7/20 0.46
NPSR1 Q6W5P4 2/20 0.45
KDM4E B2RXH2 1/20 0.45
GMNN O75496 1/20 0.45
ALDH1A1 P00352 1/20 0.45
LMNA P02545 1/20 0.45
HPGD P15428 1/20 0.45
BLM P54132 1/20 0.45
GFER P55789 1/20 0.45
PMP22 Q01453 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3669352 0.83 PDE2A (0.41) MAPK1NPSR1PTGDRFAAHCTNNB1
SCHEMBL8367478 0.81 CNR1 (0.40) ALOX15NPSR1PTGDRFAAHCTNNB1
SCHEMBL22657573 0.79 CTNNB1 (0.41) NPSR1PTGDRFAAHCTNNB1WNT3A
SCHEMBL27044834 0.78 SKP2 (0.42) MAPK1HSD17B10NPSR1ALDH1A1HPGD
SCHEMBL1971747 0.77 TAAR1 (0.53) MAPTTP53ALOX15MAPK1THPO
SCHEMBL22657669 0.77 CTNNB1 (0.43) MAPTKDM4EALDH1A1PTGDRFAAH
SCHEMBL23023195 0.77 GAA (0.51) MAPTKDM4EALDH1A1POLBSIGMAR1
SCHEMBL2663369 0.77 CTNNB1 (0.41) ALOX15NPSR1FAAHCTNNB1WNT3A
SCHEMBL1967416 0.76 SMYD3 (0.41) SMN1; SMN2PTGDRCHRM2CHRM1FAAH
SCHEMBL80920 0.76 FAAH (0.40) PTGDRFAAHCTNNB1WNT3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021011778-A1 SMALL MOLECULE INHIBITORS OF KU70/80 AND USES THEREOF ARIZONA BOARD OF REGENTS ON BEHALF OF THE UNIVERSITY OF ARIZONA (US) 2021-01-21 WO disclosed