SCHEMBL22922573

SCHEMBL22922573

Cc1cc(-c2cnc3[nH]cc(-c4ccc(C(O)N(C)C)cc4)c3c2)cc2c1N1CCN(C)CC1CC2

nearest known ligand 0.73

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAP4K1 Q92918 4/20 0.73
PIK3CG P48736 12/20 0.43
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
TNIK Q9UKE5 3/20 0.41
MAP3K11 Q16584 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29868940 0.87 MAP4K1 (0.82) MAP4K1PIK3CGTNIKMAP3K11
SCHEMBL22922379 0.87 MAP4K1 (0.82) MAP4K1PIK3CGTNIKMAP3K11
SCHEMBL29868818 0.85 MAP4K1 (1.00) MAP4K1PIK3CGCYP1A2CYP3A4CYP2D6
SCHEMBL28501865 0.85 MAP4K1 (1.00) MAP4K1PIK3CGCYP1A2CYP3A4CYP2D6
SCHEMBL29869046 0.85 MAP4K1 (1.00) MAP4K1PIK3CGCYP1A2CYP3A4CYP2D6
SCHEMBL22922558 0.85 MAP4K1 (1.00) MAP4K1PIK3CGCYP1A2CYP3A4CYP2D6
SCHEMBL22922477 0.85 MAP4K1 (1.00) MAP4K1PIK3CGCYP1A2CYP3A4CYP2D6
SCHEMBL22922557 0.85 MAP4K1 (1.00) MAP4K1PIK3CGCYP1A2CYP3A4CYP2D6
SCHEMBL22922478 0.85 MAP4K1 (1.00) MAP4K1PIK3CGCYP1A2CYP3A4CYP2D6
SCHEMBL28501867 0.85 MAP4K1 (1.00) MAP4K1PIK3CGCYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021013083-A1 TRICYCLIC COMPOUNDS AS HPK1 INHIBITOR AND THE USE THEREOF BEIGENE, LTD. (KY) 2021-01-28 WO disclosed