SCHEMBL22923656

SCHEMBL22923656

CCOC(=O)CCCN1N=C(c2ccc(N)cc2)C(C)CC1=O

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TNF P01375 6/20 0.43
FKBP1A P62942 1/20 0.38
PDE3A Q14432 3/20 0.38
PDE3B Q13370 1/20 0.38
GAA P10253 1/20 0.38
EP300 Q09472 2/20 0.37
PDE4B Q07343 3/20 0.36
NPC1 O15118 1/20 0.36
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36
TSHR P16473 1/20 0.36
RAB9A P51151 1/20 0.36
TBXAS1 P24557 1/20 0.36
PDE4A P27815 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20159196 0.80 PDE4B (0.43) PDE3APDE3BPDE4BPDE4APDE4C
SCHEMBL20159108 0.80 PDE4B (0.38) PDE3APDE3BPDE4BPDE4APDE4C
SCHEMBL22923575 0.78 PDE3A (0.43) PDE3APDE3BPDE4BPDE4APDE4C
SCHEMBL20142921 0.78 PDE4B (0.40) PDE3APDE3BPDE4BLMNAPDE4A
SCHEMBL20159457 0.78 PDE4B (0.39) PDE3APDE3BPDE4BPDE4APDE4C
SCHEMBL22923519 0.78 NAMPT (0.51)
SCHEMBL25095015 0.77 PDE4B (0.37) PDE3APDE3BPDE4BPDE4APDE4C
SCHEMBL22923624 0.77 ITGB1 (0.37) LMNAPOLBALDH1A1
SCHEMBL22923673 0.75 MEN1 (0.35) PDE3APDE3BPDE4BTSHRALDH1A1
SCHEMBL20159430 0.73 PDE4B (0.38) PDE3APDE4BPDE4APDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021013693-A1 ANTIBODY DRUG CONJUGATES (ADCS) WITH NAMPT INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2021-01-28 WO disclosed