SCHEMBL22923673

SCHEMBL22923673

CCCC(C)(C)OC(=O)NCCCN1N=C(c2ccc(N)cc2)C(C)CC1=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
MIF P14174 1/20 0.35
THRB P10828 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
MAPT P10636 1/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
HSD17B10 Q99714 1/20 0.35
DRD2 P14416 6/20 0.34
DRD3 P35462 1/20 0.34
BRD4 O60885 2/20 0.34
PDE3A Q14432 5/20 0.33
PDE4B Q07343 4/20 0.33
PDE3B Q13370 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22923610 0.82 PDE3A (0.35) DRD3PDE3APDE4BPDE3B
SCHEMBL22923576 0.80 NAMPT (0.51)
SCHEMBL22923624 0.79 ITGB1 (0.37) MEN1KMT2ATHRBKDM4EALDH1A1
SCHEMBL22923793 0.78 MIF (0.34) MEN1KMT2AMIFTHRBTDP1
SCHEMBL22923656 0.75 TNF (0.43) ALDH1A1TSHRPDE3APDE4BPDE3B
SCHEMBL20159196 0.74 PDE4B (0.43) PDE3APDE4BPDE3B
SCHEMBL20159108 0.74 PDE4B (0.38) MEN1KMT2AKDM4EALDH1A1MAPT
SCHEMBL25095015 0.73 PDE4B (0.37) MEN1KMT2AKDM4EALDH1A1MAPT
SCHEMBL20138889 0.73 PDE4B (0.41) PDE3APDE4BPDE3B
SCHEMBL20142921 0.72 PDE4B (0.40) MEN1KMT2AKDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021013693-A1 ANTIBODY DRUG CONJUGATES (ADCS) WITH NAMPT INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2021-01-28 WO disclosed