SCHEMBL22923741

SCHEMBL22923741

CCN(CC)c1ccc2cc(C(=O)OCCOCCOCCN)c(=O)oc2c1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 4/20 0.72
MEN1 O00255 8/20 0.64
MAPT P10636 8/20 0.64
KMT2A Q03164 8/20 0.64
ALDH1A1 P00352 8/20 0.64
HPGD P15428 5/20 0.64
SMN1; SMN2 Q16637 3/20 0.64
ATM Q13315 3/20 0.64
KDM4E B2RXH2 8/20 0.61
USP2 O75604 2/20 0.61
HSD17B10 Q99714 2/20 0.61
CYP1A2 P05177 1/20 0.61
CYP2C19 P33261 1/20 0.61
SLC16A3 O15427 1/20 0.61
ALOX15 P16050 1/20 0.61
SLC16A1 P53985 1/20 0.61
CYP19A1 P11511 2/20 0.52
GAA P10253 2/20 0.51
MIF P14174 1/20 0.50
PFKFB3 Q16875 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4598366 0.86 MAOB (0.80) MAOBMEN1MAPTKMT2AALDH1A1
SCHEMBL17597644 0.85 MAOB (0.79) MAOBMEN1MAPTKMT2AALDH1A1
SCHEMBL1772718 0.84 MAOB (1.00) MAOBMEN1MAPTKMT2AALDH1A1
SCHEMBL13609752 0.83 MAOB (0.72) MAOBMEN1MAPTKMT2AALDH1A1
SCHEMBL13432119 0.83 MAOB (0.76) MAOBMEN1MAPTKMT2AALDH1A1
SCHEMBL13840825 0.83 MAOB (0.76) MAOBMEN1MAPTKMT2AALDH1A1
SCHEMBL7722862 0.82 MAOB (0.74) MAOBMEN1MAPTKMT2AALDH1A1
SCHEMBL29816856 0.81 MAOB (0.80) MAOBMEN1MAPTKMT2AALDH1A1
SCHEMBL2911015 0.81 MAOB (0.80) MAOBMEN1MAPTKMT2AALDH1A1
SCHEMBL17368890 0.80 MAOB (0.71) MAOBMEN1MAPTKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021016339-A1 MODULAR CHEMICAL PROBE FOR DETECTION OF AMINO ACID CITRULLINE IN PHYSIOLOGICAL SAMPLES WISYS TECHNOLOGY FOUNDATION, INC. (US) 2021-01-28 WO disclosed