SCHEMBL22931019

SCHEMBL22931019

c1cccc(-c2ncc(-c3ccnc4[nH]ccc34)s2)c#1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 5/20 0.44
AURKB Q96GD4 3/20 0.44
IGF1R P08069 2/20 0.44
DYRK1B Q9Y463 2/20 0.44
IKBKB O14920 1/20 0.44
CHUK O15111 1/20 0.44
DAPK3 O43293 1/20 0.44
JAK2 O60674 1/20 0.44
PRKD3 O94806 1/20 0.44
MAP4K4 O95819 1/20 0.44
PAK4 O96013 1/20 0.44
CSF1R P07333 1/20 0.44
RET P07949 1/20 0.44
FGFR1 P11362 1/20 0.44
PRKACA P17612 1/20 0.44
FLT1 P17948 1/20 0.44
LTK P29376 1/20 0.44
GRK5 P34947 1/20 0.44
KDR P35968 1/20 0.44
MAP2K2 P36507 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL99315 0.79 AURKB (0.64) NUDT1AURKBIGF1RDYRK1BIKBKB
Trifluoroacetic Acid SCHEMBL98792 0.70 IKBKB (0.52) NUDT1AURKBIGF1RDYRK1BIKBKB
Trifluoroacetic Acid SCHEMBL29540629 0.70 IKBKB (0.52) NUDT1AURKBIGF1RDYRK1BIKBKB
SCHEMBL2240671 0.67 AURKB (0.71) NUDT1AURKBIGF1RDYRK1BIKBKB
SCHEMBL858198 0.67 AURKB (0.57) NUDT1AURKBIGF1RDYRK1BIKBKB
SCHEMBL4791894 0.67 AURKB (0.53) NUDT1AURKBIGF1RDYRK1BIKBKB
SCHEMBL31690444 0.67 AURKB (0.53) NUDT1AURKBIGF1RDYRK1BIKBKB
SCHEMBL29946359 0.67 AURKB (0.57) NUDT1AURKBIGF1RDYRK1BIKBKB
SCHEMBL103099 0.66 IKBKB (0.69) NUDT1AURKBIGF1RDYRK1BIKBKB
SCHEMBL29541343 0.66 IKBKB (0.69) NUDT1AURKBIGF1RDYRK1BIKBKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3466953-B1 PYRROLO[2,3-D]PYRIMIDINE DERIVATIVE AS JANUS KINASE INHIBITOR INCYTE HOLDINGS CORP (US) 2021-02-03 EP disclosed