SCHEMBL22932149

SCHEMBL22932149

C[C@H](c1ccccc1)N1CCC2(CCC(=O)NC2=O)C1

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 16/20 0.51
OPRM1 P35372 2/20 0.48
OPRD1 P41143 2/20 0.48
OPRK1 P41145 2/20 0.48
OPRL1 P41146 2/20 0.48
CYP2D6 P10635 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22932091 0.80 CRBN (0.50) CRBN
SCHEMBL22932179 0.78 CRBN (0.77) CRBN
SCHEMBL22932093 0.75 CRBN (0.45) CRBN
SCHEMBL22932062 0.73 CRBN (0.67) CRBN
SCHEMBL6840740 0.71 SIGMAR1 (0.66) OPRM1OPRD1OPRK1OPRL1CYP2D6
SCHEMBL10819303 0.70 CYP2D6 (0.60) OPRM1OPRD1OPRK1OPRL1CYP2D6
SCHEMBL28219815 0.70 CYP2D6 (0.60) OPRM1OPRD1OPRK1OPRL1CYP2D6
SCHEMBL21496463 0.70 CRBN (0.62) CRBNCYP2D6
SCHEMBL9479601 0.70 CYP2D6 (0.54) OPRM1OPRD1OPRK1OPRL1CYP2D6
SCHEMBL21496439 0.69 CRBN (0.78) CRBN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11584748-B2 Spirocyclic compounds C4 THERAPEUTICS, INC. (US) 2023-02-21 US disclosed
US-20210032245-A1 SPIROCYCLIC COMPOUNDS C4 THERAPEUTICS, INC. (US) 2021-02-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210032245-A1 SPIROCYCLIC COMPOUNDS CRBN, RBX1, XIAP CRBN 1/4885OPRM1 4739/4885OPRD1 4119/4885
US-11584748-B2 Spirocyclic compounds CRBN, RBX1, XIAP CRBN 1/4885OPRM1 4739/4885OPRD1 4119/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.