SCHEMBL22932183

SCHEMBL22932183

CS(=O)(=O)C1C=Cc2ccccc21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.36
CCL2 P13500 1/20 0.36
HTR2A P28223 2/20 0.35
HTR6 P50406 1/20 0.35
SIGMAR1 Q99720 6/20 0.33
KDM4E B2RXH2 2/20 0.33
CYP2D6 P10635 2/20 0.33
LMNA P02545 1/20 0.33
TP53 P04637 1/20 0.33
CHRM2 P08172 1/20 0.33
CYP3A4 P08684 1/20 0.33
CHRM1 P11229 1/20 0.33
DRD2 P14416 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
NFKB1 P19838 1/20 0.33
CHRM3 P20309 1/20 0.33
SLC6A2 P23975 1/20 0.33
HTR2C P28335 1/20 0.33
ADRA1A P35348 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9777608 0.83 HTR2A (0.38) BRD4CCL2HTR2AHTR6SIGMAR1
SCHEMBL30232400 0.80 HTR2A (0.39) BRD4CCL2HTR2AHTR6KDM4E
SCHEMBL2902860 0.80 HTR2A (0.39) BRD4CCL2HTR2AHTR6KDM4E
SCHEMBL31131312 0.80 HTR2A (0.35) BRD4CCL2HTR2AHTR6SIGMAR1
SCHEMBL2322179 0.80 HTR2A (0.35) BRD4CCL2HTR2AHTR6SIGMAR1
SCHEMBL14393119 0.80 HTR2A (0.35) BRD4CCL2HTR2AHTR6SIGMAR1
SCHEMBL5012228 0.80 HTR2A (0.35) BRD4CCL2HTR2AHTR6CYP2D6
SCHEMBL27512255 0.78 BRD4 (0.35) BRD4CCL2HTR2AHTR6SIGMAR1
SCHEMBL28267984 0.76 ATM (0.35) BRD4CCL2HTR2AHTR6CYP3A4
SCHEMBL28401175 0.73 SIGMAR1 (0.33) HTR2AHTR6SIGMAR1P2RX1P2RX3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115215805-A Preparation process of 2-cyanopyrimidine 上海奥萝拉医药科技有限公司 2022-10-21 CN disclosed
CN-111417409-B Pyrrolobenzodiazepine conjugates 麦迪穆有限责任公司 2022-07-08 CN disclosed
CN-113631560-A Azetidino-benzodiazepine dimers and conjugates comprising same for the treatment of cancer 麦迪穆有限责任公司 2021-11-09 CN disclosed
CN-113286617-A Pyrrolobenzodiazepine conjugates 免疫医疗有限公司 2021-08-20 CN disclosed
CN-109843335-B Pyrrolobenzodiazepine conjugates 麦迪穆有限责任公司 2021-07-30 CN disclosed
CN-112867510-A Pyrrolobenzodiazepine conjugates 免疫医疗有限公司 2021-05-28 CN disclosed
CN-111065638-B Pyrrolobenzodiazepine conjugates 麦迪穆有限责任公司 2021-04-09 CN disclosed
CN-110582505-B Pyrrolobenzodiazepine conjugates 免疫医疗有限公司 2021-04-02 CN disclosed
US-20210032449-A1 Polyethylene Copolymer and Method for Preparing Same LG CHEM, LTD. (KR) 2021-02-04 US disclosed
CN-112119082-A Pyrrolobenzodiazepines and conjugates thereof 免疫医疗有限公司 2020-12-22 CN disclosed
CN-111417409-A Pyrrolobenzodiazepine conjugates 麦迪穆有限责任公司 2020-07-14 CN disclosed
CN-111065638-A Pyrrolobenzodiazepine conjugates 麦迪穆有限责任公司 2020-04-24 CN disclosed
CN-110582505-A Pyrrolobenzodiazepine conjugates 免疫医疗有限公司 2019-12-17 CN disclosed