SCHEMBL22933197

SCHEMBL22933197

CC(=O)c1cc(-n2c(C)cc(OCc3ccccc3)cc2=O)c(C)cn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P4HTM Q9NXG6 1/20 0.45
MAOB P27338 3/20 0.44
MCHR1 Q99705 6/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
MAPK14 Q16539 1/20 0.39
GRM5 P41594 1/20 0.38
GABRA1 P14867 1/20 0.38
GABRG2 P18507 1/20 0.38
GABRB3 P28472 1/20 0.38
GABRA5 P31644 1/20 0.38
GABRA3 P34903 1/20 0.38
GABRA2 P47869 1/20 0.38
CASP3 P42574 1/20 0.38
SENP8 Q96LD8 1/20 0.38
SENP7 Q9BQF6 1/20 0.38
SENP6 Q9GZR1 1/20 0.38
ALOX5 P09917 1/20 0.38
PTGS1 P23219 1/20 0.38
PTGS2 P35354 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29963773 0.90 NPC1 (0.39) P4HTMMAOBMEN1KMT2AGRM5
SCHEMBL15311222 0.90 NPC1 (0.39) P4HTMMAOBMEN1KMT2AGRM5
SCHEMBL22933186 0.84 MAPK14 (0.43) P4HTMMAOBMCHR1MEN1KMT2A
SCHEMBL22933184 0.81 MAPK14 (0.47) MAPK14
SCHEMBL24461392 0.81 MAPKAPK5 (0.45) MAPK14
SCHEMBL29617129 0.81 MAPKAPK5 (0.45) MAPK14
SCHEMBL24926717 0.78 POLB (0.36)
SCHEMBL24759796 0.76 MAOB (0.41) MAOBMCHR1MEN1KMT2AGRM5
SCHEMBL29962567 0.76 MAOB (0.41) MAOBMCHR1MEN1KMT2AGRM5
SCHEMBL30519920 0.76 MAPKAPK5 (0.39) MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021022186-A1 DEUTERATED MK2 PATHWAY INHIBITORS AND METHODS OF USING THE SAME ACLARIS THERAPEUTICS, INC. (US) 2021-02-04 WO disclosed