SCHEMBL22938569

SCHEMBL22938569

CC(C)Nc1ccc(C(=O)O)cc1Br

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 8/20 0.59
TTR P02766 1/20 0.46
THRB P10828 3/20 0.41
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
HTT P42858 1/20 0.41
GFER P55789 1/20 0.41
PLEC Q15149 1/20 0.41
NPC1 O15118 1/20 0.41
THRA P10827 2/20 0.40
NPSR1 Q6W5P4 1/20 0.40
TPMT P51580 1/20 0.40
KDM5A P29375 1/20 0.40
PTGFR P43088 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29114266 0.80 TTR (0.50) HCAR3TTRTHRBKDM4EALDH1A1
SCHEMBL4229654 0.79 GAA (0.61) HCAR3THRBKDM4EALDH1A1GAA
SCHEMBL29114280 0.79 HCAR3 (0.59) HCAR3THRBKDM4EALDH1A1GAA
SCHEMBL31473433 0.79 GAA (0.61) HCAR3THRBKDM4EALDH1A1GAA
SCHEMBL31572042 0.79 HCAR3 (0.59) HCAR3THRBKDM4EALDH1A1GAA
SCHEMBL2617356 0.79 HCAR3 (0.59) HCAR3KDM4EALDH1A1MAPTHPGD
SCHEMBL22097623 0.77 HCAR3 (0.56) HCAR3KDM4EALDH1A1MAPTNPC1
SCHEMBL11635944 0.77 CA1 (0.57) TTRTHRBKDM4EALDH1A1GAA
SCHEMBL20604900 0.77 MAPT (0.58) HCAR3TTRTHRBKDM4EALDH1A1
SCHEMBL6187233 0.76 HCAR3 (0.55) HCAR3THRBKDM4EALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021018194-A1 HETEROCYCLIC COMPOUNDS AS BCR-ABL INHIBITORS ASCENTAGE PHARMA (SUZHOU) CO., LTD. (CN) 2021-02-04 WO disclosed