SCHEMBL2295599

SCHEMBL2295599

CN1C(=O)C(F)(F)CN(C2CCCC2)c2nc(Nc3cc(F)c(C(=O)NC4CCN(C(=O)O)CC4)cc3F)ncc21

nearest known ligand 0.77

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 18/20 0.77
BRD4 O60885 3/20 0.63
BRDT Q58F21 2/20 0.63
PLK3 Q9H4B4 4/20 0.52
PLK2 Q9NYY3 4/20 0.52
ALK Q9UM73 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1560558 0.94 PLK1 (0.87) PLK1BRD4BRDTPLK3PLK2
SCHEMBL1560401 0.91 PLK1 (0.76) PLK1BRD4BRDTPLK3PLK2
SCHEMBL1560479 0.91 PLK1 (0.75) PLK1BRD4BRDTPLK3PLK2
SCHEMBL1559960 0.91 PLK1 (0.73) PLK1BRD4BRDTPLK3PLK2
SCHEMBL1559376 0.90 PLK1 (0.74) PLK1BRD4BRDTPLK3PLK2
SCHEMBL2299583 0.90 PLK1 (0.74) PLK1BRD4BRDTALK
SCHEMBL1560553 0.87 PLK1 (0.70) PLK1BRD4BRDTPLK3PLK2
SCHEMBL1559906 0.87 PLK1 (0.67) PLK1BRD4BRDTPLK3PLK2
SCHEMBL3549236 0.87 PLK1 (0.76) PLK1BRD4BRDTPLK3PLK2
Tak-960 SCHEMBL30047124 0.87 PLK1 (1.00) PLK1BRD4BRDTPLK3PLK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8003785-B2 Halo-substituted pyrimidodiazepines TAKEDA PHARMACEUTICAL COMPANY LIMITED (US) 2011-08-23 US disclosed