SCHEMBL22958360

SCHEMBL22958360

Cc1ccc2c(c1Cl)NC(=O)CC2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 3/20 0.40
CYP11B2 P19099 3/20 0.40
CYP1A2 P05177 1/20 0.40
NPC1 O15118 1/20 0.39
MAPK13 O15264 1/20 0.39
MAPK12 P53778 1/20 0.39
MAPK11 Q15759 1/20 0.39
MAPK14 Q16539 1/20 0.39
PKM P14618 8/20 0.39
CA9 Q16790 1/20 0.39
SRD5A1 P18405 1/20 0.36
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
AHR P35869 1/20 0.36
CYP19A1 P11511 2/20 0.35
ALDH1A1 P00352 1/20 0.35
CES1 P23141 1/20 0.35
HTR1A P08908 1/20 0.35
DRD2 P14416 1/20 0.35
HTR2A P28223 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27148030 0.81 NPC1 (0.41) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL30893045 0.81 NPC1 (0.41) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL434004 0.74 NPC1 (0.50) CYP11B1CYP11B2NPC1MAPK13MAPK12
SCHEMBL12559751 0.74 CYP11B1 (0.46) CYP11B1CYP11B2CYP1A2NPC1MAPK13
Hydrochloric Acid SCHEMBL29961795 0.73 NPC1 (0.48) CYP11B1CYP11B2NPC1MAPK13MAPK12
SCHEMBL10911499 0.73 KDM4E (0.39) ALDH1A1HTR2ATP53
SCHEMBL12559620 0.73 CES1 (0.43) CYP11B1CYP11B2CYP1A2PKMAHR
SCHEMBL24427466 0.71 PKM (0.41) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL14494366 0.71 PDE3B (0.46) CYP11B1CYP11B2CYP1A2NPC1MAPK13
SCHEMBL30893019 0.71 SRD5A1 (0.40) NPC1MAPK13MAPK12MAPK11MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3772513-A1 SHP2 INHIBITORS C.N.C.C.S. S.c.a.r.l. Collezione Nazionale Dei Composti Chimici e Centro Screening (IT) 2021-02-10 EP disclosed