SCHEMBL22965729

SCHEMBL22965729

CNNc1c(N)cccc1Br

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.37
TSHR P16473 2/20 0.37
PIK3CA P42336 1/20 0.37
ALDH1A1 P00352 3/20 0.33
TDP1 Q9NUW8 2/20 0.33
CD44 P16070 1/20 0.33
HPGD P15428 1/20 0.33
HSD17B10 Q99714 1/20 0.33
ALOX15 P16050 1/20 0.32
CASP1 P29466 1/20 0.32
CASP7 P55210 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
MAPK13 O15264 1/20 0.32
MAPK12 P53778 1/20 0.32
MAPK11 Q15759 1/20 0.32
MAPK14 Q16539 1/20 0.32
BACE1 P56817 2/20 0.31
TAAR1 Q96RJ0 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29799761 0.84 CYP3A4 (0.39) CYP3A4TSHRPIK3CAALDH1A1TDP1
SCHEMBL933021 0.84 CYP3A4 (0.39) CYP3A4TSHRPIK3CAALDH1A1TDP1
Hydrochloric Acid SCHEMBL15158274 0.83 CYP3A4 (0.37) CYP3A4TSHRPIK3CAALDH1A1TDP1
SCHEMBL32676372 0.77 MAPT (0.37) CYP3A4TSHRPIK3CAALDH1A1TDP1
SCHEMBL2018207 0.75 KDM4E (0.36) CYP3A4TSHRPIK3CAALDH1A1TDP1
SCHEMBL4259819 0.75 HSD17B10 (0.36) CYP3A4TSHRPIK3CAALDH1A1TDP1
SCHEMBL31204396 0.75 KDM4E (0.36) CYP3A4TSHRPIK3CAALDH1A1TDP1
SCHEMBL4628755 0.72 HDAC1 (0.48) ALDH1A1HPGDHSD17B10
SCHEMBL5149864 0.71 HDAC1 (0.47) ALDH1A1HPGDHSD17B10
SCHEMBL11901586 0.71 MAPT (0.50) CYP3A4TSHRALDH1A1TDP1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021026375-A1 FUSED BICYCLIC COMPOUNDS FOR THE TREATMENT OF PAIN ALKERMES, INC. (US) 2021-02-11 WO disclosed