SCHEMBL5149864

SCHEMBL5149864

CC(=O)Nc1c(N)cccc1Br.[Fe]

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.47
ALDH1A1 P00352 4/20 0.43
RXFP1 Q9HBX9 1/20 0.41
CYP1A2 P05177 2/20 0.41
EGFR P00533 1/20 0.40
POLB P06746 2/20 0.39
KCNJ11 Q14654 1/20 0.38
HSD17B10 Q99714 3/20 0.38
NAPRT Q6XQN6 1/20 0.38
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
CA9 Q16790 2/20 0.38
HDAC3 O15379 1/20 0.38
HDAC2 Q92769 1/20 0.38
KDM4E B2RXH2 2/20 0.38
MAPT P10636 1/20 0.38
GLA P06280 1/20 0.38
HPGD P15428 1/20 0.38
RAB9A P51151 1/20 0.37
CA12 O43570 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4628755 0.98 HDAC1 (0.48) HDAC1ALDH1A1RXFP1CYP1A2EGFR
SCHEMBL21807836 0.85 RXFP1 (0.48) ALDH1A1RXFP1CYP1A2EGFRPOLB
SCHEMBL22158291 0.79 RXFP1 (0.44) ALDH1A1RXFP1CYP1A2EGFRPOLB
SCHEMBL9187652 0.78 ALDH1A1 (0.50) HDAC1ALDH1A1RXFP1CYP1A2EGFR
SCHEMBL12247210 0.78 ALDH1A1 (0.50) HDAC1ALDH1A1CYP1A2POLBHSD17B10
SCHEMBL11022909 0.78 HDAC1 (0.49) HDAC1ALDH1A1CYP1A2POLBKCNJ11
SCHEMBL5149869 0.77 HDAC1 (0.37) HDAC1ALDH1A1CYP1A2CA1CA2
SCHEMBL16240385 0.76 HDAC1 (0.48) HDAC1ALDH1A1RXFP1CYP1A2EGFR
SCHEMBL3412158 0.76 HDAC1 (0.48) HDAC1ALDH1A1CYP1A2POLBHSD17B10
SCHEMBL601500 0.76 HDAC1 (0.72) HDAC1ALDH1A1CYP1A2HDAC3HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1608627-A4 BICYCLIC ANILIDE SPIROHYDANTOIN CGRP RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2007-08-01 EP disclosed
EP-1608627-A2 BICYCLIC ANILIDE SPIROHYDANTOIN CGRP RECEPTOR ANTAGONISTS Merck & Co. Inc. (US) 2005-12-28 EP disclosed
WO-2004082605-A2 BICYCLIC ANILIDE SPIROHYDANTOIN CGRP RECEPTOR ANTAGONISTS MERCK & CO. INC. (US) 2004-09-30 WO disclosed